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Found 23 with Last Name = 'prachyawarakorn' and Initial = 'v'
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50000541((+-)-1-(1-Benzo[b]thien-2-ylethyl)-1-hydroxyurea |...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant 5-LOX assessed as reduction in leukotriene B4 synthesis using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510095(CHEMBL4465694)
Affinity DataIC50:  400nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  590nMAssay Description:Inhibition of AChE activityMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510097(CHEMBL4553272)
Affinity DataIC50:  800nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510098(CHEMBL4515706)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant 5-LOX assessed as reduction in leukotriene B4 synthesis using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510098(CHEMBL4515706)
Affinity DataIC50:  900nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510095(CHEMBL4465694)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant 5-LOX assessed as reduction in leukotriene B4 synthesis using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510097(CHEMBL4553272)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant 5-LOX assessed as reduction in leukotriene B4 synthesis using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510096(ARAHYPIN-5)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human recombinant 5-LOX assessed as reduction in leukotriene B4 synthesis using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM35440(ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510097(CHEMBL4553272)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM50182887(1-(3,4-dimethoxy-benzyl)-6,7-dimethoxy-2-methyl-3,...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of AChE activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510095(CHEMBL4465694)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM50182888((6,7-dimethoxyisoquinolin-1-yl)(2-methoxyphenyl)me...)
Affinity DataIC50:  6.94E+3nMAssay Description:Inhibition of AChE activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM50182890((6,7-dimethoxyisoquinolin-1-yl)(3,4-dimethoxypheny...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of AChE activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510099(CHEMBL4517895)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510096(ARAHYPIN-5)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510098(CHEMBL4515706)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510096(ARAHYPIN-5)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM14754(1-[(3,4-dimethoxyphenyl)methyl]-6,7-dimethoxy-isoq...)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of AChE activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50510099(CHEMBL4517895)
Affinity DataIC50:  3.55E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as reduction in PGE2 production using arachidonic acid substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed