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Found 262 with Last Name = 'rai' and Initial = 'v'
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585913(CHEMBL5093295)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585914(CHEMBL5079273)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585912(CHEMBL5075486)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585909(CHEMBL5089996)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585910(CHEMBL5094012)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585911(CHEMBL5093969)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585918(CHEMBL5078567)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585915(CHEMBL5082151)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585919(CHEMBL5090584)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585920(CHEMBL5092524)
Affinity DataKi:  271nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585916(CHEMBL5085238)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585917(CHEMBL5091270)
Affinity DataKi:  705nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to human 5-HT5ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT2BR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT2AR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT1DR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT1BR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT1AR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT2CR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585922(CHEMBL5079940)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585901(CHEMBL3459329)
Affinity DataKi:  1.14E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585901(CHEMBL3459329)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585905(CHEMBL5087322)
Affinity DataKi:  1.28E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585905(CHEMBL5087322)
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585903(CHEMBL5074821)
Affinity DataKi:  2.08E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585903(CHEMBL5074821)
Affinity DataKi:  2.09E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585902(CHEMBL5092728)
Affinity DataKi:  2.13E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585902(CHEMBL5092728)
Affinity DataKi:  2.14E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585904(CHEMBL5093652)
Affinity DataKi:  2.88E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585904(CHEMBL5093652)
Affinity DataKi:  2.88E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of FLT3 ITD mutant (unknown orgin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50604641(CHEMBL5183674)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of FLT3 ITD mutant (unknown orgin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344869(1'-pentyl-6H-spiro[benzofuro[6,5-d][1,3]dioxole-7,...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50587891(CHEMBL5181237 | US11814388, Compound 4)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of EGFR (unknown origin) using Poly(Glu, Tyr) as substrate incubated for 45 mins in presence of ATP by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of wild type FLT3 (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50604641(CHEMBL5183674)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of wild type FLT3 (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344821(10-hydroxymethyl-5-imino-(2S)-12,13-dioxa-4,6-diaz...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50604642(CHEMBL5206333)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of FLT3 ITD mutant (unknown orgin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445731(CHEMBL3104392)
Affinity DataIC50:  12nMAssay Description:Inhibition of SCD1 in human HepG2 cells using radiolabeled stearic acid as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50486734(CHEMBL5289303)
Affinity DataIC50:  12nMAssay Description:Inhibition of VEGFR2 (unknown origin) at 25 nM using Poly(Glu, Tyr) as substrate by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50486735(CHEMBL5274698)
Affinity DataIC50:  14nMAssay Description:Inhibition of VEGFR2 (unknown origin) at 25 nM using Poly(Glu, Tyr) as substrate by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM50604642(CHEMBL5206333)
Affinity DataIC50:  14nMAssay Description:Inhibition of wild type FLT3 (unknown origin) by ADP-glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445732(CHEMBL3104401)
Affinity DataIC50:  14nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445734(CHEMBL3104405)
Affinity DataIC50:  15nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445728(CHEMBL3104407)
Affinity DataIC50:  18nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445738(CHEMBL3104406)
Affinity DataIC50:  20nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445726(CHEMBL3104390)
Affinity DataIC50:  20nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344834(3-(benzo[d][1,3]dioxol-5-yl)-1-(2-cyclopropylethyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445737(CHEMBL3104395)
Affinity DataIC50:  24nMAssay Description:Inhibition of SCD1 in mouse liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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