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Found 71 with Last Name = 'rastagar' and Initial = 'a'
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  9nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182908(1-((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenyla...)
Affinity DataIC50:  9nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182891(CHEMBL205798 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  12nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182900(CHEMBL381604 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  12nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182893((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamin...)
Affinity DataIC50:  13nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182891(CHEMBL205798 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  13nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182908(1-((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenyla...)
Affinity DataIC50:  15nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50261965(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182906(CHEMBL205045 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  17nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182892(CHEMBL206003 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  21nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262113(2-((5-chloro-1H-indol-3-yl)methyl)-7-(cyclopropylm...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182895(1-((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenyla...)
Affinity DataIC50:  23nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262115(2-((5-chloro-1H-indol-3-yl)methyl)-7-(cyclopropylm...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50215445(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262011(5-(2-((5-chloro-1H-indol-3-yl)methyl)-7-(cycloprop...)
Affinity DataIC50:  27nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182898(CHEMBL206782 | methyl 5-(3-(2-(4-(4-(3-fluorobenzy...)
Affinity DataIC50:  29nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182910(CHEMBL205966 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  30nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182898(CHEMBL206782 | methyl 5-(3-(2-(4-(4-(3-fluorobenzy...)
Affinity DataIC50:  31nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262060(2-((5-chloro-1H-indol-3-yl)methyl)-7-(cyclopropylm...)
Affinity DataIC50:  31nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182907(CHEMBL381080 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  32nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182912(3-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino...)
Affinity DataIC50:  32nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182900(CHEMBL381604 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  32nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182904((5-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamin...)
Affinity DataIC50:  33nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262163(2-((5-chloro-1-methyl-1H-indol-3-yl)methyl)-7-(cyc...)
Affinity DataIC50:  33nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262114(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropylme...)
Affinity DataIC50:  34nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262012(5-(2-((5-chloro-1H-indol-3-yl)methyl)-7-(cycloprop...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182910(CHEMBL205966 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  36nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262061(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropylme...)
Affinity DataIC50:  37nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182892(CHEMBL206003 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  38nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50261964(2-(2-((5-chloro-1H-indol-3-yl)methyl)-7-(cycloprop...)
Affinity DataIC50:  38nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182893((6-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamin...)
Affinity DataIC50:  40nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182896(CHEMBL205235 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  42nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182915(5-(2-(1H-pyrazol-3-yl)ethynyl)-N-(4-(3-fluorobenzy...)
Affinity DataIC50:  42nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182896(CHEMBL205235 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  44nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50261966(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50:  44nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182899(CHEMBL208358 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  45nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182904((5-(2-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamin...)
Affinity DataIC50:  47nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182907(CHEMBL381080 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  50nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50261912(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropylme...)
Affinity DataIC50:  51nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182897(CHEMBL207247 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  52nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50262013(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50:  55nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182906(CHEMBL205045 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  55nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50261913(2-((5-chloro-1-methyl-1H-indol-3-yl)methyl)-7-(cyc...)
Affinity DataIC50:  57nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182913(CHEMBL205765 | N-(6-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  59nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50261911(3-(3-chloro-5-(methylsulfonyl)furan-2-yl)-2-((6-ch...)
Affinity DataIC50:  59nMAssay Description:Inhibition of Helicobacter pylori MurIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182897(CHEMBL207247 | N-(3-(2-(4-(4-(3-fluorobenzyloxy)-3...)
Affinity DataIC50:  60nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182901(CHEMBL207869 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  60nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182894(CHEMBL204625 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  63nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50182915(5-(2-(1H-pyrazol-3-yl)ethynyl)-N-(4-(3-fluorobenzy...)
Affinity DataIC50:  66nMAssay Description:Inhibition of ErbB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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