Affinity DataKi: 62nMAssay Description:Inhibition of Trypanosoma cruzi squalene synthaseMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of Trypanosoma cruzi squalene synthaseMore data for this Ligand-Target Pair
Affinity DataKi: 133nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 297nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 516nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 598nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 641nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 733nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 802nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 808nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 815nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 847nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Competitive inhibition of recombinant human KLK1 expressed in baculovirus/insect cell expression system using Abz-KLRSSKQ-EDDnp peptide as substrate ...More data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.81E+3nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.79E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.73E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.76E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.40E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.22E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.45E+4nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant carbonic anhydrase-2-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant carbonic anhydrase-1-mediated CO2 hydration by stopped-flow assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 0.331nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 0.479nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 0.490nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 0.575nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 0.794nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 0.955nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 1.29nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 2.51nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 2.82nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 2.88nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 3.63nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 3.63nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 4.27nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 4.57nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 5.13nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro (Ufrj)
Curated by ChEMBL
Affinity DataIC50: 5.75nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Tested for inhibitory potency against rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair