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Found 228 with Last Name = 'rush' and Initial = 'ts'
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173235((S)-2-{4'-[(5-Bromo-4-methoxy-benzofuran-2-carbony...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  0.430nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  0.600nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173236((S)-2-{4'-[(5-Bromo-benzofuran-2-carbonyl)-amino]-...)
Affinity DataIC50:  0.610nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  0.660nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173236((S)-2-{4'-[(5-Bromo-benzofuran-2-carbonyl)-amino]-...)
Affinity DataIC50:  0.910nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50:  0.980nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170304((S)-2-{4'-[(5-Amino-benzofuran-2-carbonyl)-amino]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173220((S)-2-{4'-[(5-Chloro-4-methoxy-3-methyl-benzofuran...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173218((S)-2-{4'-[(5-Iodo-4-methoxy-3-methyl-benzofuran-2...)
Affinity DataIC50:  2.10nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170299((S)-3-Methyl-2-{4'-[([1,2,3]thiadiazole-4-carbonyl...)
Affinity DataIC50:  2.10nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170289((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173223((S)-2-(4'-(5-bromo-4-methoxy-3-methylbenzofuran-2-...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173223((S)-2-(4'-(5-bromo-4-methoxy-3-methylbenzofuran-2-...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50297236((S)-2-(4'-(4-ethyl-3-methylbenzofuran-2-carboxamid...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170295((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM24043((2R)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173229((S)-2-{4'-[(5-Cyano-4-methoxy-3-methyl-benzofuran-...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173224((S)-2-{4'-[(5-Bromo-3-methyl-benzofuran-2-carbonyl...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173237((S)-2-{4'-[(5-Acetyl-4-hydroxy-3-methyl-benzofuran...)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173221((R)-2-{4'-[(5-Bromo-4-methoxy-3-methyl-benzofuran-...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170288((S)-2-{4'-[(5-Benzenesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170296((S)-2-{4'-[(4-Benzyloxy-benzofuran-2-carbonyl)-ami...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50297239((S)-2-(4'-(4-cyano-3-methylbenzofuran-2-carboxamid...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173228((S)-2-{4'-[(5-Ethyl-4-methoxy-3-methyl-benzofuran-...)
Affinity DataIC50:  3.80nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50297229((S)-2-(4'-(4-amino-3-methylbenzofuran-2-carboxamid...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM24047((2R)-3-methyl-2-[(4-{4-[(3-methyl-1-benzofuran-2-y...)
Affinity DataIC50:  4.40nMpH: 7.5 T: 2°CAssay Description:A continuous assay was used in which the substrate is a synthetic peptide containing a fluorescent group (7-methoxycoumarin), which is quenched by en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170286((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM24043((2R)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50297235((S)-2-(4'-(3,4-dimethylbenzofuran-2-carboxamido)bi...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173222((S)-2-{4'-[(4-methoxy-3,5-dimethyl-benzofuran-2-ca...)
Affinity DataIC50:  4.90nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50:  4.90nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  5nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50173226((S)-3-Methyl-2-{4'-[(3-methyl-benzofuran-2-carbony...)
Affinity DataIC50:  5.90nMAssay Description:Inhibitory concentration against MMP-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50297240((S)-2-(4'-(4-ethynyl-3-methylbenzofuran-2-carboxam...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50297225((S)-2-(4'-(4-hydroxy-3-methylbenzofuran-2-carboxam...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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