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Found 54 with Last Name = 'rushmore' and Initial = 't'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391916(CHEMBL2147556)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391923(CHEMBL2147566)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391920(CHEMBL2147562)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391913(CHEMBL2147553)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391917(CHEMBL2147557)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391919(CHEMBL2147561)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391924(CHEMBL2147567)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391925(CHEMBL2147569)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391918(CHEMBL2147558)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251022(3-(4-hydroxy-3,5-diiodobenzoyl)-2-propyl-4H-chrome...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273790(6-Bromo-N-(naphthalen-2-yl)-2-(pyridin-4-yl)quinol...)
Affinity DataKi:  9nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391922(CHEMBL2147564)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273447(6,8-Dimethyl-N-(naphthalen-2-yl)-2-(pyridin-4-yl)q...)
Affinity DataKi:  11nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273788(6-Chloro-N-(naphthalen-2-yl)-2-(pyridin-4-yl)quino...)
Affinity DataKi:  12nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391914(CHEMBL2147554)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50158460((3,5-dibromo-4-hydroxyphenyl)(2-ethyl-1-benzofuran...)
Affinity DataKi:  19nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251021(2-ethyl-3-(4-hydroxy-3,5-diiodobenzoyl)-4H-chromen...)
Affinity DataKi:  23nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273785(CHEMBL456181 | N-(Naphthalen-2-yl)-2-(pyridin-4-yl...)
Affinity DataKi:  33nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391921(CHEMBL2147563)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251020(3-(4-hydroxy-3,5-diiodobenzoyl)-2-methyl-4H-chrome...)
Affinity DataKi:  41nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251136(3-(3,5-diiodo-4-methoxybenzoyl)-2-propyl-4H-chrome...)
Affinity DataKi:  44.3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391926(CHEMBL2147572)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273444(CHEMBL463976 | N-Phenyl-2-(pyridin-4-yl)quinoline-...)
Affinity DataKi:  100nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50232842(3-(3,5-dibromo-4-hydroxybenzoyl)-2-ethyl-4H-chrome...)
Affinity DataKi:  101nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273393(CHEMBL514730 | N-(Naphthalen-1-ylmethyl)-2-(pyridi...)
Affinity DataKi:  113nMAssay Description:Inhibition of purified CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273393(CHEMBL514730 | N-(Naphthalen-1-ylmethyl)-2-(pyridi...)
Affinity DataKi:  125nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273394(CHEMBL463577 | N-(Naphthalen-1-ylmethyl)-2-(pyridi...)
Affinity DataKi:  152nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391915(CHEMBL2147555)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391928(CHEMBL2147629)
Affinity DataKi: >400nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50391927(CHEMBL2147573)
Affinity DataKi: >400nMAssay Description:Displacement of [3H]-dexamethasone from human full length GR expressed in insect Sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251122(3-(4-hydroxybenzoyl)-2-propyl-4H-chromen-4-one | C...)
Affinity DataKi:  656nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273786(CHEMBL456182 | N-(Naphthalen-2-yl)-2-(pyridin-3-yl...)
Affinity DataKi:  1.15E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273819(CHEMBL456185 | N-(Naphthalen-1-yl)-2-(pyridin-3-yl...)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273820(CHEMBL515841 | N-(Naphthalen-1-yl)-2-(pyridin-2-yl...)
Affinity DataKi:  1.32E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251121(2-ethyl-3-(4-hydroxybenzoyl)-4H-chromen-4-one | CH...)
Affinity DataKi:  1.42E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273789(6-Chloro-N-(naphthalen-2-yl)-2-(pyridin-3-yl)quino...)
Affinity DataKi:  1.89E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251135(3-(4-methoxybenzoyl)-2-propyl-4H-chromen-4-one | C...)
Affinity DataKi:  3.12E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273446(CHEMBL513115 | N-Phenyl-2-(pyridin-2-yl)quinoline-...)
Affinity DataKi:  3.47E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273782((2-(Pyridin-4-yl)quinolin-4-yl)(4-(pyrrolidin-1-yl...)
Affinity DataKi:  3.67E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273445(CHEMBL464389 | N-Phenyl-2-(pyridin-3-yl)quinoline-...)
Affinity DataKi:  4.06E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251119(2-ethyl-3-isonicotinoyl-4H-chromen-4-one | CHEMBL4...)
Affinity DataKi:  4.87E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251123(3-(4-methoxybenzoyl)-2-methyl-4H-chromen-4-one | C...)
Affinity DataKi:  5.93E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251134(2-ethyl-3-(4-methoxybenzoyl)-4Hchromen-4-one | CHE...)
Affinity DataKi:  6.48E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50251120(3-(4-hydroxybenzoyl)-2-methyl-4H-chromen-4-one | C...)
Affinity DataKi:  6.74E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273448(6,8-Dimethyl-N-(naphthalen-2-yl)-2-(pyridin-3-yl)q...)
Affinity DataKi:  8.55E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273712(CHEMBL457021 | Piperidin-1-yl(2-(pyridin-3-yl)quin...)
Affinity DataKi:  9.74E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273711(CHEMBL511703 | Piperidin-1-yl(2-(pyridin-4-yl)quin...)
Affinity DataKi:  9.94E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273392(CHEMBL456998 | N-(Naphthalen-2-yl)-2-(pyridin-2-yl...)
Affinity DataKi:  1.07E+4nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273787(6,8-Dimethyl-N-(naphthalen-2-yl)-2-(pyridin-2-yl)q...)
Affinity DataKi: >2.06E+4nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50273713(CHEMBL511852 | Piperidin-1-yl(2-(pyridin-2-yl)quin...)
Affinity DataKi:  2.36E+4nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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