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Found 193 with Last Name = 'sabatino' and Initial = 'm'
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593468(CHEMBL5199803)
Affinity DataIC50:  0.190nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593464(CHEMBL5184399)
Affinity DataIC50:  0.260nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593462(CHEMBL5178058)
Affinity DataIC50:  0.330nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593471(CHEMBL5195371)
Affinity DataIC50:  0.390nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593476(CHEMBL5191405)
Affinity DataIC50:  0.670nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593472(CHEMBL5174813)
Affinity DataIC50:  0.710nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)
Affinity DataIC50:  0.740nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593473(CHEMBL5207726)
Affinity DataIC50:  0.75nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593466(CHEMBL5187253)
Affinity DataIC50:  0.760nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  0.890nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  0.890nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593474(CHEMBL5203282)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50180684(4-OHT | Afimoxifene | TamoGel)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593475(CHEMBL5178110)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50180684(4-OHT | Afimoxifene | TamoGel)
Affinity DataIC50:  3.60nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593463(CHEMBL5209099)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593477(CHEMBL5194045)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593467(CHEMBL5196340)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593469(CHEMBL5181808)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593470(CHEMBL5187730)
Affinity DataIC50:  39nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593472(CHEMBL5174813)
Affinity DataIC50:  43nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593465(CHEMBL5198828)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593475(CHEMBL5178110)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593476(CHEMBL5191405)
Affinity DataIC50:  67nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593474(CHEMBL5203282)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593469(CHEMBL5181808)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50126143(Epacadostat | INCB-024360)
Affinity DataIC50:  72nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50126143(Epacadostat | INCB-024360)
Affinity DataIC50:  72nMAssay Description:Inhibition of human IDO1More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593470(CHEMBL5187730)
Affinity DataIC50:  74nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593462(CHEMBL5178058)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593471(CHEMBL5195371)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593466(CHEMBL5187253)
Affinity DataIC50:  86nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593464(CHEMBL5184399)
Affinity DataIC50:  98nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593472(CHEMBL5174813)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at ERalpha in human MCF7 cells assessed as downregulation of ERalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50180684(4-OHT | Afimoxifene | TamoGel)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593476(CHEMBL5191405)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593475(CHEMBL5178110)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593474(CHEMBL5203282)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593473(CHEMBL5207726)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593472(CHEMBL5174813)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593471(CHEMBL5195371)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593470(CHEMBL5187730)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593469(CHEMBL5181808)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593468(CHEMBL5199803)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593466(CHEMBL5187253)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593464(CHEMBL5184399)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at progesterone receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593462(CHEMBL5178058)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at ERalpha in human MCF7 cells assessed as downregulation of ERalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593464(CHEMBL5184399)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at ERalpha in human MCF7 cells assessed as downregulation of ERalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593466(CHEMBL5187253)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at ERalpha in human MCF7 cells assessed as downregulation of ERalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Kragujevac

Curated by ChEMBL
LigandPNGBDBM50593468(CHEMBL5199803)
Affinity DataIC50: >100nMAssay Description:Antagonist activity at ERalpha in human MCF7 cells assessed as downregulation of ERalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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