Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.07nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.99nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.49nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Affinity DataKi: 3.71nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.82nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.93nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.23nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.93nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.92nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.68nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.57nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.62nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 14.6nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 14.9nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 15.4nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 15.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17.6nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 18.8nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 21.1nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23.8nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 30.9nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 32.7nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 34.1nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 35.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 36.7nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 37.6nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 37.8nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 37.8nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 38.1nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 38.2nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 38.6nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 44.4nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 46.1nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 47.3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 52.8nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 55.2nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 62.9nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 63.4nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 64.1nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 69.3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
B.V. Patel Pharmaceutical Education And Research Development
Curated by ChEMBL
Affinity DataKi: 75.4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair