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Found 48 with Last Name = 'sackett' and Initial = 'dl'
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM18129((2S)-2-amino-3-(4-hydroxyphenyl)propanoic acid | L...)
Affinity DataKi:  2.50E+4nM ΔG°:  -27.3kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36556(3-Azidotyrosine)
Affinity DataKi:  2.00E+5nM ΔG°:  -22.0kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36555(3-Aminotyrosine)
Affinity DataKi:  2.00E+5nM ΔG°:  -22.0kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36557(3-Formyltyrosine)
Affinity DataKi:  3.00E+5nM ΔG°:  -20.9kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36554(3-Nitrotyrosine)
Affinity DataKi:  4.00E+5nM ΔG°:  -20.2kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36558(4-Aminophenylalanine)
Affinity DataKi: >4.00E+6nM ΔG°: >-14.2kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475544(CHEMBL372120)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81747(Chembridge No 9067250, Class 1, 8)
Affinity DataIC50:  5.20E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81744(Oryzalin Analogue, 3)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81745(Oryzalin Analogue, 4)
Affinity DataIC50:  6.60E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475546(CHEMBL382519)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81746(Chembridge No 7992831, 5)
Affinity DataIC50:  1.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475541(CHEMBL196754)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81746(Chembridge No 7992831, 5)
Affinity DataIC50:  3.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81743(Oryzalin, 1)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81744(Oryzalin Analogue, 3)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475545(CHEMBL381416)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50131995((E)-3-(4-hydroxybenzylidene)indolin-2-one | 3-(4-H...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475543(CHEMBL382323)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475542(CHEMBL378162)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81743(Oryzalin, 1)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81745(Oryzalin Analogue, 4)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81747(Chembridge No 9067250, Class 1, 8)
Affinity DataIC50:  5.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81748(Chembridge No 7946770, Class 1, 9)
Affinity DataIC50:  5.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81753(Chembridge No 9035165, Class 2, 13)
Affinity DataIC50:  6.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81752(Chembridge No 9035650, Class 2, 12)
Affinity DataIC50:  6.10E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81753(Chembridge No 9035165, Class 2, 13)
Affinity DataIC50:  6.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81751(Chembridge No 9041709, Class 2, 11)
Affinity DataIC50:  6.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81749(Chembridge No 7960631, Class 1, 10)
Affinity DataIC50:  6.40E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81752(Chembridge No 9035650, Class 2, 12)
Affinity DataIC50:  6.60E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81748(Chembridge No 7946770, Class 1, 9)
Affinity DataIC50:  6.70E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81749(Chembridge No 7960631, Class 1, 10)
Affinity DataIC50:  6.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81751(Chembridge No 9041709, Class 2, 11)
Affinity DataIC50:  6.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81750(Chembridge No 9063043, Class 1, 17)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81750(Chembridge No 9063043, Class 1, 17)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81754(Chembridge No 7944934, Class 2, 16)
Affinity DataIC50:  7.10E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81757(Chembridge No 9049411, Class 4, 15)
Affinity DataIC50:  7.20E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81756(Chembridge No 9056942, Class 3, 7)
Affinity DataIC50:  7.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81758(Chembridge No 9044486, Class 4, 6)
Affinity DataIC50:  8.10E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81755(Chembridge No 9026860, Class 3, 14)
Affinity DataIC50:  8.90E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81754(Chembridge No 7944934, Class 2, 16)
Affinity DataIC50:  9.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81757(Chembridge No 9049411, Class 4, 15)
Affinity DataIC50:  1.07E+5nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81755(Chembridge No 9026860, Class 3, 14)
Affinity DataIC50:  1.11E+5nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81758(Chembridge No 9044486, Class 4, 6)
Affinity DataIC50:  1.20E+5nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81756(Chembridge No 9056942, Class 3, 7)
Affinity DataIC50:  1.40E+5nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed