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maximum 50k data
Found 117 with Last Name = 'sackur' and Initial = 'c'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215802(CHEMBL233559 | methyl 4-(6-(diisopentylcarbamoyl)-...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215802(CHEMBL233559 | methyl 4-(6-(diisopentylcarbamoyl)-...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215807(CHEMBL392092 | N,N-diisopentyl-2-(4-methoxybenzoyl...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215807(CHEMBL392092 | N,N-diisopentyl-2-(4-methoxybenzoyl...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215841(2-(4-benzoylphenylamino)-N,N-diisopentyl-3-(3-(pip...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215841(2-(4-benzoylphenylamino)-N,N-diisopentyl-3-(3-(pip...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215816(2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215816(2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215844(CHEMBL232161 | N,N-diisopentyl-2-(4-phenoxyphenyla...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215844(CHEMBL232161 | N,N-diisopentyl-2-(4-phenoxyphenyla...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215813(CHEMBL395226 | N,N-diisopentyl-2-(4-nitrophenylami...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215813(CHEMBL395226 | N,N-diisopentyl-2-(4-nitrophenylami...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215836(CHEMBL233757 | N,N-diisopentyl-3-(3-(piperidin-1-y...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215836(CHEMBL233757 | N,N-diisopentyl-3-(3-(piperidin-1-y...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215820(2-(benzo[b]thiophen-2-yl)-N,N-diisopentyl-3-(3-(pi...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215820(2-(benzo[b]thiophen-2-yl)-N,N-diisopentyl-3-(3-(pi...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215801(CHEMBL391664 | N,N-diisopentyl-2-(1-methyl-1H-indo...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215801(CHEMBL391664 | N,N-diisopentyl-2-(1-methyl-1H-indo...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215828(CHEMBL233758 | N,N-diisopentyl-2-(4-(methylcarbamo...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215828(CHEMBL233758 | N,N-diisopentyl-2-(4-(methylcarbamo...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215812(2-(4-acetamidophenylamino)-N,N-diisopentyl-3-(3-(p...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215812(2-(4-acetamidophenylamino)-N,N-diisopentyl-3-(3-(p...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215800(2-(4-acetylbenzyl)-N,N-diisopentyl-3-(3-(piperidin...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215800(2-(4-acetylbenzyl)-N,N-diisopentyl-3-(3-(piperidin...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215823(CHEMBL232584 | N,N-diisopentyl-3-(3-(piperidin-1-y...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215823(CHEMBL232584 | N,N-diisopentyl-3-(3-(piperidin-1-y...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215846(2-(3-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215846(2-(3-acetylphenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215805(2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pyrr...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215805(2-(4-acetylphenylamino)-N,N-diisopentyl-3-(3-(pyrr...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215815(CHEMBL429943 | N,N-diisopentyl-2-(4-methoxyphenyla...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215815(CHEMBL429943 | N,N-diisopentyl-2-(4-methoxyphenyla...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215839(2-(biphenyl-4-ylamino)-3-(3-piperidin-1-yl-propyl)...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215839(2-(biphenyl-4-ylamino)-3-(3-piperidin-1-yl-propyl)...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215831(2-(4-acetylbenzylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215831(2-(4-acetylbenzylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215835(2-(4-carbamoylphenylamino)-N,N-diisopentyl-3-(3-(p...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215835(2-(4-carbamoylphenylamino)-N,N-diisopentyl-3-(3-(p...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215804(2-(1H-indol-3-yl)-N,N-diisopentyl-3-(3-(piperidin-...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215804(2-(1H-indol-3-yl)-N,N-diisopentyl-3-(3-(piperidin-...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215845(CHEMBL430165 | N,N-diisopentyl-2-(phenylamino)-3-(...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215845(CHEMBL430165 | N,N-diisopentyl-2-(phenylamino)-3-(...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215829(2-(4-bromophenylamino)-N,N-diisopentyl-3-(3-(piper...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215829(2-(4-bromophenylamino)-N,N-diisopentyl-3-(3-(piper...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215833(2-(4-acetylphenylamino)-3-(3-(diethylamino)propyl)...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215833(2-(4-acetylphenylamino)-3-(3-(diethylamino)propyl)...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215852(2-(4-fluorophenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215852(2-(4-fluorophenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215811(2-(4-chlorophenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50215811(2-(4-chlorophenylamino)-N,N-diisopentyl-3-(3-(pipe...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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