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Found 103 with Last Name = 'sahu' and Initial = 'nu'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123830(4,5-dibromo-N'-(4-chlorobenzylidene)-1-methyl-...)
Affinity DataKi:  2.10E+3nM ΔG°:  -33.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123825(4,5-dibromo-N'-[(4-fluorophenyl)methylidene]-1...)
Affinity DataKi:  2.40E+3nM ΔG°:  -33.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123833(4,5-dibromo-N'-(2,4-dichlorobenzylidene)-1-met...)
Affinity DataKi:  2.60E+3nM ΔG°:  -33.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123832(4,5-dibromo-N'-(4-methoxybenzylidene)-1-methyl...)
Affinity DataKi:  2.90E+3nM ΔG°:  -32.9kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123823(4,5-dibromo-N'-[(2,4-dichlorophenyl)methyliden...)
Affinity DataKi:  3.10E+3nM ΔG°:  -32.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123831(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1-me...)
Affinity DataKi:  3.40E+3nM ΔG°:  -32.5kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123828(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1-met...)
Affinity DataKi:  3.90E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123820(4,5-dibromo-N'-[(4-chlorophenyl)methylidene]-1...)
Affinity DataKi:  3.90E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123824(4,5-dibromo-N'-(2-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  4.70E+3nM ΔG°:  -31.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123815(4,5-dibromo-N'-(4-fluorobenzylidene)-1H-pyrrol...)
Affinity DataKi:  5.10E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123818(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1Hpyr...)
Affinity DataKi:  5.20E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123829(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1-me...)
Affinity DataKi:  6.10E+3nM ΔG°:  -31.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123822(4,5-dibromo-N'-(4-methoxybenzylidene)-1Hpyrrol...)
Affinity DataKi:  6.55E+3nM ΔG°:  -30.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123826(4,5-dibromo-1-methyl-N'-(4-nitrobenzylidene)-1...)
Affinity DataKi:  6.90E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123827(4,5-dibromo-N'-(4-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  7.10E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123814(4,5-dibromo-N'-(2-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  8.90E+3nM ΔG°:  -30.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123823(4,5-dibromo-N'-[(2,4-dichlorophenyl)methyliden...)
Affinity DataKi:  9.40E+3nM ΔG°:  -29.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123821(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1Hpy...)
Affinity DataKi:  1.13E+4nM ΔG°:  -29.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123828(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1-met...)
Affinity DataKi:  1.23E+4nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123820(4,5-dibromo-N'-[(4-chlorophenyl)methylidene]-1...)
Affinity DataKi:  1.25E+4nM ΔG°:  -29.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123833(4,5-dibromo-N'-(2,4-dichlorobenzylidene)-1-met...)
Affinity DataKi:  1.29E+4nM ΔG°:  -29.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123827(4,5-dibromo-N'-(4-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  1.33E+4nM ΔG°:  -29.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123832(4,5-dibromo-N'-(4-methoxybenzylidene)-1-methyl...)
Affinity DataKi:  1.38E+4nM ΔG°:  -28.9kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123816(4,5-dibromo-N'-(4-nitrobenzylidene)-1H-pyrrole...)
Affinity DataKi:  1.44E+4nM ΔG°:  -28.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123817(4,5-dibromo-N'-(4-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  1.59E+4nM ΔG°:  -28.5kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123819(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1Hpy...)
Affinity DataKi:  1.73E+4nM ΔG°:  -28.3kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123829(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1-me...)
Affinity DataKi:  2.04E+4nM ΔG°:  -27.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123818(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1Hpyr...)
Affinity DataKi:  2.05E+4nM ΔG°:  -27.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123822(4,5-dibromo-N'-(4-methoxybenzylidene)-1Hpyrrol...)
Affinity DataKi:  2.12E+4nM ΔG°:  -27.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123831(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1-me...)
Affinity DataKi:  2.17E+4nM ΔG°:  -27.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123824(4,5-dibromo-N'-(2-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  2.28E+4nM ΔG°:  -27.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123815(4,5-dibromo-N'-(4-fluorobenzylidene)-1H-pyrrol...)
Affinity DataKi:  2.45E+4nM ΔG°:  -27.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123821(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1Hpy...)
Affinity DataKi:  2.61E+4nM ΔG°:  -27.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123830(4,5-dibromo-N'-(4-chlorobenzylidene)-1-methyl-...)
Affinity DataKi:  2.69E+4nM ΔG°:  -27.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123814(4,5-dibromo-N'-(2-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  3.78E+4nM ΔG°:  -26.3kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123825(4,5-dibromo-N'-[(4-fluorophenyl)methylidene]-1...)
Affinity DataKi:  3.81E+4nM ΔG°:  -26.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123826(4,5-dibromo-1-methyl-N'-(4-nitrobenzylidene)-1...)
Affinity DataKi:  4.05E+4nM ΔG°:  -26.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123817(4,5-dibromo-N'-(4-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  4.26E+4nM ΔG°:  -26.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123819(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1Hpy...)
Affinity DataKi:  4.48E+4nM ΔG°:  -25.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123816(4,5-dibromo-N'-(4-nitrobenzylidene)-1H-pyrrole...)
Affinity DataKi:  6.63E+4nM ΔG°:  -24.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Nmims University

Curated by ChEMBL
LigandPNGBDBM50491188(CHEMBL151430)
Affinity DataIC50:  6nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531537(CHEMBL4474709)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531532(CHEMBL4462468)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531536(CHEMBL194094)
Affinity DataIC50:  1.97E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531535(CHEMBL4470070)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531539(CHEMBL4283519)
Affinity DataIC50:  3.37E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531534(CHEMBL4289201)
Affinity DataIC50:  3.58E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531531(CHEMBL4540332)
Affinity DataIC50:  3.75E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531543(CHEMBL4538625)
Affinity DataIC50:  4.28E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50531533(CHEMBL4589531)
Affinity DataIC50:  4.74E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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