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Found 770 with Last Name = 'saito' and Initial = 'r'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490612(CHEMBL2337603)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490602(CHEMBL2338047)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490637(CHEMBL2338049)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490621(CHEMBL2338048)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490599(CHEMBL2337596)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490592(CHEMBL2337595)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490625(CHEMBL2338034)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490611(CHEMBL2337604)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490600(CHEMBL2337602)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490606(CHEMBL2338039)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490635(CHEMBL2337593)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490638(CHEMBL2338051)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490609(CHEMBL2338032)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490631(CHEMBL2338050)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490601(CHEMBL2337592)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490590(CHEMBL2338053)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118202(6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490632(CHEMBL2338045)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490604(CHEMBL2338042)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490619(CHEMBL2338055)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490624(CHEMBL2338035)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490630(CHEMBL2338052)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490633(CHEMBL2338033)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490593(CHEMBL2338043)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490620(CHEMBL2338054)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490597(CHEMBL2337591)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490622(CHEMBL2338044)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490615(CHEMBL2337594)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490613(CHEMBL2337598)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490607(CHEMBL2338037)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490595(CHEMBL2337605)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118204(6-(4-benzoylphenylcarbonyloxy)-8-(tert-butyl)-12,1...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118201(6-(4-benzoylbenzyloxy)-8-(tert-butyl)-12,17-dihydr...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118194(8-(tert-butyl)-12,17-dihydroxy-16-methyl-6-[4-(3-t...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490614(CHEMBL2337597)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490610(CHEMBL2338031)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490626(CHEMBL2337608)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490591(CHEMBL2337590)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490616(CHEMBL2337589)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490627(CHEMBL2337607)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490629(CHEMBL2337606)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490603(CHEMBL2338046)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490605(CHEMBL2338041)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490608(CHEMBL2338036)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118203(8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-6-[4-(...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50490617(CHEMBL2337587)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]WIN35428 from human recombinant DAT transfected in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118195(3'-(tert-butyl)-4,9',14'-trihydroxy-2-methoxy-10'-...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118196(6-(4-benzoylbenzyloxy)-8-(tert-butyl)-9,12,17-trih...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118200(6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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