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Found 68 with Last Name = 'sakai-moritani' and Initial = 'y'
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209900(3-(({7-[amino(imino)methyl]-2-naphthyl}methyl)-{1-...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209891(CHEMBL390266 | [(((E)-3-{3-[amino(imino)methyl]phe...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209893(7-({[1-(2,5-dimethoxy-benzenesulfonyl)-piperidin-4...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209895(CHEMBL244221 | N-({7-[amino(imino)methyl]-2-naphth...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209899(3-(((E)-3-{3-[amino(imino)methyl]phenyl}prop-2-en-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209904(CHEMBL244436 | [(({7-[amino(imino)methyl]-2-naphth...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209920(7-({[1-(5-chloro-2-methoxy-benzenesulfonyl)-piperi...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209915(7-({[1-(3-chloro-benzenesulfonyl)-piperidin-4-yl]-...)
Affinity DataIC50:  49nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209896(7-({methanesulfonyl-[1-(2-methoxy-5-methyl-benzene...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209914(7-({[1-(2,5-dichloro-benzenesulfonyl)-piperidin-4-...)
Affinity DataIC50:  65nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM31459(CHEMBL224485 | substituted biphenyl derivative, 21)
Affinity DataIC50:  89nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209905(7-{[(methylsulfonyl)(1-pyridin-4-ylpiperidin-4-yl)...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209908(7-({[1-(2,5-dichloro-thiophene-3-sulfonyl)-piperid...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197327(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209911(7-({[1-(3-cyano-benzenesulfonyl)-piperidin-4-yl]-m...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197325(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209916(7-({[1-(3,4-dichloro-benzenesulfonyl)-piperidin-4-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209917(7-({[1-(biphenyl-3-sulfonyl)-piperidin-4-yl]-metha...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209894(7-({methanesulfonyl-[1-(toluene-3-sulfonyl)-piperi...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197331(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-({...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197330(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209912(7-({[1-(2-chloro-benzenesulfonyl)-piperidin-4-yl]-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209921(7-({[1-(2,3-dichloro-benzenesulfonyl)-piperidin-4-...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197324(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209901(7-{[{1-[(2,5-dimethoxyphenyl)sulfonyl]piperidin-4-...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197326(2'-(3-carbamoyl-phenylcarbamoyl)-4-isobutylcarbamo...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209918(7-({[1-(3-fluoro-benzenesulfonyl)-piperidin-4-yl]-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209897(7-{[(1-benzenesulfonyl-piperidin-4-yl)-methanesulf...)
Affinity DataIC50:  850nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197329(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  860nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM31459(CHEMBL224485 | substituted biphenyl derivative, 21)
Affinity DataIC50:  880nMAssay Description:Inhibition of human Fxa by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209903(7-({methanesulfonyl-[1-(toluene-2-sulfonyl)-piperi...)
Affinity DataIC50:  950nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197340(2'-({[4-(aminomethyl)phenyl]amino}carbonyl)-4-({[(...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209919(7-({[1-(4-chloro-benzenesulfonyl)-piperidin-4-yl]-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209892(7-({[1-(3-chloro-benzyl)-piperidin-4-yl]-methanesu...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197336(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209909(7-({[1-(3-cyano-benzyl)-piperidin-4-yl]-methanesul...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197341(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197333(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-[(...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197334(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-[(...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197332(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}carb...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197338(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197335(2'-(3-Carbamoyl-phenylcarbamoyl)-4-isobutylcarbamo...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197339(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197328(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209895(CHEMBL244221 | N-({7-[amino(imino)methyl]-2-naphth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209891(CHEMBL390266 | [(((E)-3-{3-[amino(imino)methyl]phe...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209900(3-(({7-[amino(imino)methyl]-2-naphthyl}methyl)-{1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209902(7-[(methanesulfonyl-piperidin-4-yl-amino)-methyl]-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50209893(7-({[1-(2,5-dimethoxy-benzenesulfonyl)-piperidin-4...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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