Affinity DataKi: 3nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.40E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7.10E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:The NLRP3 inflammasome inhibitory activity of test compounds were evaluated CM the basis of the inhibitory activity of the IL-1β, production in ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.980nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 6(Homo sapiens (Human))
Daiichi Sankyo
Curated by ChEMBL
Daiichi Sankyo
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human TRPC6 expressed in HEK293 cells assessed as decrease in intracellular calcium level after 24 hrs by Fluo-4 dye-based FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Human SGLT1-stably-expressing cell lines were seeded at 5×104 cells/well on BioCoat™ Poly-D-Lysine 96 well plate with Lid (Becton, Dickinson and Comp...More data for this Ligand-Target Pair