Affinity DataKi: 0.200nMAssay Description:Agonistic activity at DRD3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Antagonistic activity at human DRD3 receptor by filtration binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Antagonistic activity at rat DRD3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-pentazocin from the Sigma1 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-pentazocin from the Sigma1 receptorMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-DTG from the Sigma2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Agonistic activity at DRD2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-pentazocin from the Sigma1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15.8nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15.8nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair