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Found 263 with Last Name = 'salis' and Initial = 'a'
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Redx Pharma

Curated by ChEMBL
LigandPNGBDBM50463770(CHEMBL4238919)
Affinity DataIC50:  5nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanC-like protein 2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50041087(CHEMBL3355910)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of ABA binding to LANCL2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Redx Pharma

Curated by ChEMBL
LigandPNGBDBM50463771(CHEMBL4250651)
Affinity DataIC50:  10nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Redx Pharma

Curated by ChEMBL
LigandPNGBDBM50226181((3R,4S,5R,6R)-5-hydroxy-6-(4-hydroxy-3-(4-hydroxy-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase ATPase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Redx Pharma

Curated by ChEMBL
LigandPNGBDBM50463770(CHEMBL4238919)
Affinity DataIC50:  25nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase ATPase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600005(CHEMBL5195268)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600003(CHEMBL5201228)
Affinity DataIC50:  55nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Redx Pharma

Curated by ChEMBL
LigandPNGBDBM50463771(CHEMBL4250651)
Affinity DataIC50:  59nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase ATPase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Redx Pharma

Curated by ChEMBL
LigandPNGBDBM50226181((3R,4S,5R,6R)-5-hydroxy-6-(4-hydroxy-3-(4-hydroxy-...)
Affinity DataIC50:  85nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600006(CHEMBL5172158)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600007(CHEMBL5182200)
Affinity DataIC50:  105nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553249(CHEMBL4743440)
Affinity DataIC50:  200nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600004(CHEMBL5184104)
Affinity DataIC50:  220nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553247(CHEMBL4764598)
Affinity DataIC50:  300nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600009(CHEMBL5177076)
Affinity DataIC50:  340nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600008(CHEMBL5198597)
Affinity DataIC50:  460nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553247(CHEMBL4764598)
Affinity DataIC50:  500nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553248(CHEMBL4787847)
Affinity DataIC50:  800nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553249(CHEMBL4743440)
Affinity DataIC50:  800nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553249(CHEMBL4743440)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553250(CHEMBL4786331)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase using relaxed pBR322 as substrate incubated for 30 mins by ethidium bromide staining based gel electro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553248(CHEMBL4787847)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600011(CHEMBL5205047)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600007(CHEMBL5182200)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600003(CHEMBL5201228)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600010(CHEMBL5184352)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553250(CHEMBL4786331)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase IV using kDNA as substrate incubated for 30 mins by ethidium bromide staining based gel electrophor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553249(CHEMBL4743440)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600018(CHEMBL5199405)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600013(CHEMBL5194618)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553247(CHEMBL4764598)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553247(CHEMBL4764598)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600014(CHEMBL5172094)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600012(CHEMBL5190832)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553247(CHEMBL4764598)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553249(CHEMBL4743440)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553249(CHEMBL4743440)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553247(CHEMBL4764598)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600017(CHEMBL5195721)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600003(CHEMBL5201228)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553250(CHEMBL4786331)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553250(CHEMBL4786331)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600015(CHEMBL5206169)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50536777(CHEMBL4526887)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human ERG channel by automated patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451276(CHEMBL4217987)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553250(CHEMBL4786331)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of Nav1.5 (unknown origin) by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451275(CHEMBL4205716)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50553248(CHEMBL4787847)
Affinity DataIC50:  2.26E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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