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Found 37 with Last Name = 'samanta' and Initial = 'h'
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184633(6-(3,4-dichlorophenyl)-2-hydroxy-4-oxohex-2-enoic ...)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM23399(4-{1-[(4-fluorophenyl)methyl]-1H-pyrrol-2-yl}-2,4-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM107693((2Z)-4-(5-chloro-1H-indol-3-yl)-2-hydroxy-4-oxobut...)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184626(6-(2-chlorophenyl)-2,4,6-trioxohexanoic acid | CHE...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM23399(4-{1-[(4-fluorophenyl)methyl]-1H-pyrrol-2-yl}-2,4-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM107693((2Z)-4-(5-chloro-1H-indol-3-yl)-2-hydroxy-4-oxobut...)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184626(6-(2-chlorophenyl)-2,4,6-trioxohexanoic acid | CHE...)
Affinity DataIC50:  600nMAssay Description:Inhibition of HIV1 recombinant integrase in pre-integration complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184632(6-(naphthalen-1-yl)-2,4,6-trioxohexanoic acid | CH...)
Affinity DataIC50:  600nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184626(6-(2-chlorophenyl)-2,4,6-trioxohexanoic acid | CHE...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184630(6-biphenyl-4-yl-2,4,6-trioxo-hexanoic acid | CHEMB...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184635(6-(2-fluorophenyl)-2,4,6-trioxohexanoic acid | CHE...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184624(6-(2-methoxyphenyl)-2,4,6-trioxohexanoic acid | CH...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184625(6-(2-bromophenyl)-2-hydroxy-4-oxohex-2-enoic acid ...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184623(2,4,6-trioxo-6-(2-(trifluoromethyl)phenyl)hexanoic...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184638(6-(naphthalen-2-yl)-2,4,6-trioxohexanoic acid | CH...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184631(6-(2-(benzyloxy)phenyl)-2,4,6-trioxohexanoic acid ...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184637(6-(3-chlorophenyl)-2,4,6-trioxohexanoic acid | CHE...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184622(6-(2-chlorophenyl)-2-hydroxy-4-oxohex-2-enoic acid...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184622(6-(2-chlorophenyl)-2-hydroxy-4-oxohex-2-enoic acid...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184628(2-hydroxy-4-oxo-6-phenylhex-2-enoic acid | CHEMBL2...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184634(2,4,6-trioxo-6-phenylhexanoic acid | CHEMBL448424)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184636(2,4,6-trioxo-6-(pyridin-2-yl)hexanoic acid | CHEMB...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184627(1-(2-chlorophenyl)-5-(1H-tetrazol-5-yl)pentane-1,3...)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184639(1-(1-(4-fluorobenzyl)-1H-pyrrol-2-yl)-3-(1H-tetraz...)
Affinity DataIC50: >1.25E+5nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50184621(2,4,6-trioxo-6-(pyridin-3-yl)hexanoic acid | CHEMB...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of HIV1 recombinant integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450016(CHEMBL4163247)
Affinity DataKd:  49nMAssay Description:Binding affinity to HIV1 gag polyprotein V370A mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450015(Bms-955176 | GSK-3532795)
Affinity DataKd:  34nMAssay Description:Binding affinity to HIV1 gag polyprotein delta V370 mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450016(CHEMBL4163247)
Affinity DataKd:  259nMAssay Description:Binding affinity to HIV1 gag polyprotein delta V370 mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50538906(CHEMBL4649761)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of HIV-1 integrase strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50538907(CHEMBL4637079)
Affinity DataEC50: >6.40E+4nMAssay Description:Inhibition of HIV-1 integrase strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450015(Bms-955176 | GSK-3532795)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to HIV1 gag polyprotein V370A mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450016(CHEMBL4163247)
Affinity DataKd:  15nMAssay Description:Binding affinity to HIV1 gag polyprotein V362I mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450015(Bms-955176 | GSK-3532795)
Affinity DataKd:  4.30nMAssay Description:Binding affinity to HIV1 gag polyprotein V362I mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50450015(Bms-955176 | GSK-3532795)
Affinity DataKd:  3.20nMAssay Description:Binding affinity to wild type HIV1 gag polyprotein containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50450015(Bms-955176 | GSK-3532795)
Affinity DataKd:  98nMAssay Description:Binding affinity to HIV1 gag polyprotein A364V mutant containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50538908(CHEMBL4642318)
Affinity DataEC50:  9.30E+3nMAssay Description:Inhibition of HIV-1 integrase strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50450016(CHEMBL4163247)
Affinity DataKd:  5.40nMAssay Description:Binding affinity to wild type HIV1 gag polyprotein containing viral like particleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed