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Found 141 with Last Name = 'samaras' and Initial = 's'
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50:  0.0400nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168170(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.0460nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182367(4-(2-(4-fluorophenyl)-7-(piperidin-4-yl)H-imidazo[...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374578(CHEMBL401749)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374594(CHEMBL444009)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182359(CHEMBL379059 | N-benzyl-4-(7-((dimethylamino)methy...)
Affinity DataIC50:  0.0810nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195444(2-(ethyl((2-(4-fluorophenyl)-3-(2-((S)-1-phenyleth...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195435(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)py...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195439(CHEMBL221636 | N-((2-(4-fluorophenyl)-3-(2-((S)-1-...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182355(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.130nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195446(CHEMBL222158 | N-((2-(4-fluorophenyl)-3-(2-((S)-1-...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182358(4-(2-(4-fluorophenyl)-7-((methylamino)methyl)H-imi...)
Affinity DataIC50:  0.150nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168185(4-[2-(3-Bromo-4-fluoro-phenyl)-5-(1-methyl-piperid...)
Affinity DataIC50:  0.150nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182361(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.150nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195441(CHEMBL220598 | N-ethyl-N-((2-(4-fluorophenyl)-3-(2...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374591(CHEMBL255128)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195433(CHEMBL221689 | N-((2-(4-fluorophenyl)-3-(2-((S)-1-...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195437((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)pyrimi...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171694((R)-5-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-py...)
Affinity DataIC50:  0.160nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182356(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374587(CHEMBL272573)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182363(4-(7-(aminomethyl)-2-(4-fluorophenyl)H-imidazo[1,2...)
Affinity DataIC50:  0.180nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168208(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374588(CHEMBL255381)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195443((3-(2-(benzyloxy)pyrimidin-4-yl)-2-(4-fluorophenyl...)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168187(4-{2-(4-Fluoro-phenyl)-5-[1-(1-methyl-azetidin-2-y...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168202(2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168206(4-[5-(1-Ethyl-piperidin-4-yl)-2-(4-fluoro-phenyl)-...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374592(CHEMBL271922)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168192(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.320nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195434(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374580(CHEMBL271638)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50183915((5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-y...)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374590(CHEMBL406910)
Affinity DataIC50:  0.360nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171685(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.380nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374593(CHEMBL429745)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171698(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171707(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.410nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168190(4-[2-(3-Chloro-4-fluoro-phenyl)-5-(1-methyl-piperi...)
Affinity DataIC50:  0.440nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171705(1-Benzyloxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50195447(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.470nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171699((S)-1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-py...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168176(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.530nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168176(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.530nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171695((R)1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyr...)
Affinity DataIC50:  0.560nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171688(1-Ethoxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-...)
Affinity DataIC50:  0.590nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171702(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.660nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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