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Found 467 with Last Name = 'samatar' and Initial = 'aa'
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50:  0.800nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50094464(CHEMBL3590107 | US10525036, Example SCH772984 | US...)
Affinity DataIC50:  1nMAssay Description:Inhibition of ERK2 (unknown origin) preincubated for 45 mins followed by substrate addition measured after 0.5 hrs by IMAP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50094464(CHEMBL3590107 | US10525036, Example SCH772984 | US...)
Affinity DataIC50:  1nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458811(CHEMBL4209570)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579208(CHEMBL4867107)
Affinity DataIC50:  2nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103295(US8546404, 462)
Affinity DataIC50:  2.10nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM103295(US8546404, 462)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579222(CHEMBL4861383)
Affinity DataIC50:  2.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518531(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518527(2-Alyl-6-((2′,3′-dihydro-1′H-spi...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518526(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518538(2-Allyl-6-((2-(2-hydroxyethyl)-1,2,3,4-tetrahydroi...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103292(US8546404, 1729 | US8546404, 469)
Affinity DataIC50:  2.5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM34531(US8546404, 459)
Affinity DataIC50:  2.5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579228(CHEMBL4867211)
Affinity DataIC50:  2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103292(US8546404, 1729 | US8546404, 469)
Affinity DataIC50:  2.5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518540(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579214(CHEMBL4856035)
Affinity DataIC50:  2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579225(CHEMBL4874546)
Affinity DataIC50:  2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518530(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579218(CHEMBL4876612)
Affinity DataIC50:  2.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579223(CHEMBL4853285)
Affinity DataIC50:  3.10nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579224(CHEMBL4861351)
Affinity DataIC50:  3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579227(CHEMBL4847705)
Affinity DataIC50:  3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579221(CHEMBL4866800)
Affinity DataIC50:  3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579216(CHEMBL4865963)
Affinity DataIC50:  3.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579213(CHEMBL4853973)
Affinity DataIC50:  3.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579220(CHEMBL4868683)
Affinity DataIC50:  3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579219(CHEMBL4857841)
Affinity DataIC50:  3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50:  3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)
Affinity DataIC50:  3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579215(CHEMBL4861168)
Affinity DataIC50:  4.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103293(US8546404, 480)
Affinity DataIC50:  4.80nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579211(CHEMBL4871803)
Affinity DataIC50:  4.80nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM103293(US8546404, 480)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458805(CHEMBL4206960)
Affinity DataIC50:  5nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458806(CHEMBL4205192)
Affinity DataIC50:  5nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103296(US8546404, 622)
Affinity DataIC50:  5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579212(CHEMBL4879157)
Affinity DataIC50:  5.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50461920(CHEMBL4225841)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458802(CHEMBL4215228)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458802(CHEMBL4215228)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579210(CHEMBL4853185)
Affinity DataIC50:  5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579210(CHEMBL4853185)
Affinity DataIC50:  5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50461917(CHEMBL4225054)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458807(CHEMBL4216900)
Affinity DataIC50:  6nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetWee1-like protein kinase(Homo sapiens (Human))
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579209(CHEMBL4874090)
Affinity DataIC50:  6.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM103297(US8546404, 613)
Affinity DataIC50:  7nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM103297(US8546404, 613)
Affinity DataIC50:  7nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50458803(CHEMBL4213970)
Affinity DataIC50:  7nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
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