Compile Data Set for Download or QSAR
maximum 50k data
Found 26 with Last Name = 'sambucini' and Initial = 's'
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of flag-tagged HDAC3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataIC50:  1nMAssay Description:Inhibition of flag-tagged HDAC4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  1nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of flag-tagged HDAC4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of HDAC4 catalytic domain expressed in HEK293 cells by Biomol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of flag-tagged HDAC3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of flag-tagged HDAC4 expressed in HEK293 cells by Biomol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  4nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM50377931(CHEMBL1791402)
Affinity DataIC50:  88nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM50377931(CHEMBL1791402)
Affinity DataIC50:  152nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260229(4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human CKIdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  510nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260228(CHEMBL489344 | N-methyl-4-(2-(piperidin-4-yl)-5-(3...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human CKIalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260229(4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human CKIalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260228(CHEMBL489344 | N-methyl-4-(2-(piperidin-4-yl)-5-(3...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human CKIdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260229(4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260228(CHEMBL489344 | N-methyl-4-(2-(piperidin-4-yl)-5-(3...)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260229(4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260228(CHEMBL489344 | N-methyl-4-(2-(piperidin-4-yl)-5-(3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260229(4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...)
Affinity DataIC50:  1.66E+5nMAssay Description:Inhibition of human JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260229(4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-im...)
Affinity DataIC50:  1.75E+5nMAssay Description:Inhibition of human JNK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260228(CHEMBL489344 | N-methyl-4-(2-(piperidin-4-yl)-5-(3...)
Affinity DataIC50:  3.85E+5nMAssay Description:Inhibition of human JNK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti

Curated by ChEMBL
LigandPNGBDBM50260228(CHEMBL489344 | N-methyl-4-(2-(piperidin-4-yl)-5-(3...)
Affinity DataIC50:  4.04E+5nMAssay Description:Inhibition of human JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed