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Found 46 with Last Name = 'sammons' and Initial = 'r'
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281993(CHEMBL287334 | Trisodium salt of (3R,4S,5R)-5-Carb...)
Affinity DataKi:  1.50E+3nMAssay Description:Dissociation constant of the compound was calculated for E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392849(CHEMBL2151190 | US9073941, 612)
Affinity DataIC50:  500nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392855(CHEMBL1969923)
Affinity DataIC50:  630nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392849(CHEMBL2151190 | US9073941, 612)
Affinity DataIC50:  700nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392849(CHEMBL2151190 | US9073941, 612)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392855(CHEMBL1969923)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392856(CHEMBL1981814)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392856(CHEMBL1981814)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392854(CHEMBL1980140)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392857(CHEMBL1492532)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392860(CHEMBL2151286)
Affinity DataIC50:  7.80E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392858(FURALTADONE)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392859(CHEMBL2151285)
Affinity DataIC50:  1.45E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392860(CHEMBL2151286)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392859(CHEMBL2151285)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  4.10E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  4.30E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  5.80E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281993(CHEMBL287334 | Trisodium salt of (3R,4S,5R)-5-Carb...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281990(CHEMBL33426 | Trisodium salt of (3R,4S,5R)-5-(1-Ca...)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  1.97E+5nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.52E+5nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.95E+5nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281995(CHEMBL284334 | Disodium salt of 3-Phosphonooxy-cyc...)
Affinity DataIC50:  7.50E+6nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281987(2-(3-Carboxy-cyclohex-2-enyloxy)-malonic acid | CH...)
Affinity DataIC50:  1.50E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281994(CHEMBL430544 | Disodium salt of (3R,4R,5R)-5-(1-Ca...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281345((3R,4R,5R)-5-Carboxymethoxy-3,4-dihydroxy-cyclohex...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281986(3-Phosphonomethylene-cyclohex-1-enecarboxylic acid...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281991(3-Phosphonomethoxy-cyclohex-1-enecarboxylic acid |...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281989(CHEMBL285416 | Sodium; (3-carboxy-5,6-dihydroxy-cy...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281992(CHEMBL32407 | Disodium salt of 3-Phosphonomethyl-c...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281996(2-(3-Carboxy-cyclohex-2-enyl)-malonic acid | CHEMB...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281998((3R,4S,5R)-3,4,5-trihydroxycyclohex-1-ene-1-carbox...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281997(3-Phosphonomethylene-cyclohex-1-enecarboxylic acid...)
Affinity DataIC50: >9.00E+7nMAssay Description:Inhibition of E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281990(CHEMBL33426 | Trisodium salt of (3R,4S,5R)-5-(1-Ca...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity of the compound was determined against E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
Target3-phosphoshikimate 1-carboxyvinyltransferase(Escherichia coli (strain K12))
TBA

Curated by ChEMBL
LigandPNGBDBM50281988(CHEMBL32352 | Sodium salt of (3R,4S,5R)-4,5-Dihydr...)
Affinity DataKd:  7.00E+3nMAssay Description:Inhibitory activity of the compound was evaluated against E. coli EPSP(5-enolpyruvyl-shikimate-3-phosphate) SynthaseMore data for this Ligand-Target Pair
In DepthDetails Article