TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 794nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 6.31E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 7.94E+5nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human 20S proteasome beta5 subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human 20S immunoproteasome beta-1i subunit using (Ac-PAL)2R110 as substrate preincubated for 2 hrs followed by substrate addition and m...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human 20S immunoproteasome beta-1i subunit using (Ac-PAL)2R110 as substrate preincubated for 2 hrs followed by substrate addition and m...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human 20S proteasome beta5 subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of 20S immunoproteasome beta-5i subunit in human PBMC using Ac-ANW-luciferin substrate preincubated for 2 hrs followed by substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human 20S proteasome beta5 subunit using Suc-LLVY-AMC as substrate preincubated for 2 hrs followed by substrate addition and measured a...More data for this Ligand-Target Pair