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Found 35 with Last Name = 'sangshetti' and Initial = 'jn'
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50468271(CHEMBL4290134)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50612120(CHEMBL5275705)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50505333(CHEMBL4437173)
Affinity DataIC50:  7nMAssay Description:Inhibition of TNKS1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50019166(CHEMBL336718)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))TBA
LigandPNGBDBM50505333(CHEMBL4437173)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of human recombinant TNKS2 expressed in Escherichia coli assessed as inhibition at 20 uM measured after 48 hrs by fluorescence based analy...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50188337(CHEMBL2058057)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))TBA
LigandPNGBDBM50511566(CHEMBL4448872)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant TNKS2More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50612121(CHEMBL5277753)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50511566(CHEMBL4448872)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant TNKS1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50612117(CHEMBL5270676)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50612118(CHEMBL3431396)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50612119(CHEMBL5267866)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant full length TNKS1 (1030 to 1317 residues) expressed in Escherichia coli assessed as inhibition by fluorescence based ...More data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  990nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179406(CHEMBL3814850)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570427(CHEMBL4864715)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570429(CHEMBL4878037)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179404(CHEMBL3814663)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179409(CHEMBL3814475)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570428(CHEMBL4870551)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570432(CHEMBL4849502)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179402(CHEMBL3814494)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179429(CHEMBL3814111)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179410(CHEMBL3815111)
Affinity DataIC50:  2.28E+4nMAssay Description:Inhibition of Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179408(CHEMBL3814560)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570430(CHEMBL4855587)
Affinity DataIC50:  2.64E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179400(CHEMBL3814987)
Affinity DataIC50:  2.78E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179411(CHEMBL3815003)
Affinity DataIC50:  2.83E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179407(CHEMBL3814606)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179412(CHEMBL3814562)
Affinity DataIC50:  3.35E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179405(CHEMBL3814751)
Affinity DataIC50:  3.46E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570431(CHEMBL4869150)
Affinity DataIC50:  3.99E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179399(CHEMBL3814600)
Affinity DataIC50:  4.25E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University

Curated by ChEMBL
LigandPNGBDBM50570433(CHEMBL4853443)
Affinity DataIC50:  4.84E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179401(CHEMBL3814164)
Affinity DataIC50:  5.08E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Y.B. Chavan College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50179428(CHEMBL3814974)
Affinity DataIC50:  5.12E+4nMAssay Description:Inhibition of NiCl2 stabilized Escherichia coli NCIM-2931 peptide deformylase using N-formyl-Met-Ala as substrate incubated for 30 mins by spectropho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed