Compile Data Set for Download or QSAR
maximum 50k data
Found 104 with Last Name = 'sano' and Initial = 'h'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85790(Salmon MCH)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85789([Phe13,Tyr19]MCH)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85789([Phe13,Tyr19]MCH)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85788(MCH | hMCH)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85790(Salmon MCH)
Affinity DataKi:  437nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145539((2S,4R)-2,4-Dihydroxy-6-[2-[(R)-1-((R)-5-hydroxy-1...)
Affinity DataIC50:  0.5nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145538((S)-1-Benzyl-5-((R)-2-{(R)-4-[2-[(3S,5R)-3,5-dihyd...)
Affinity DataIC50:  1.90nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062251(CHEMBL285263 | trisodium 5-[2-benzo[d][1,3]dioxol-...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062250(CHEMBL36407 | trisodium 5-[2-benzo[d][1,3]dioxol-5...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062249(CHEMBL285434 | trisodium 5-[2-benzo[d][1,3]dioxol-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062249(CHEMBL285434 | trisodium 5-[2-benzo[d][1,3]dioxol-...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of Farnesyltransferase in competitive manner with respect to FPP (farnesyl diphosphate) at 0.6 microM FPP and 0.36 microM Ras peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062252(CHEMBL36339 | trisodium 5-[2-benzo[d][1,3]dioxol-5...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062248(CHEMBL36515 | trisodium 5-[2-benzo[d][1,3]dioxol-5...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062249(CHEMBL285434 | trisodium 5-[2-benzo[d][1,3]dioxol-...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of Farnesyltransferase in competitive manner with respect to FPP (farnesyl diphosphate) at 0.6 microM FPP and 3.6 microM Ras peptide.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062256(CHEMBL284073 | trisodium 5-[2-benzo[d][1,3]dioxol-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145540((S)-5-((R)-2-{(R)-4-[2-[(3S,5R)-3,5-Dihydroxy-2-me...)
Affinity DataIC50:  10nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062258(2-{[((E)-2-Benzo[1,3]dioxol-5-yl-5-benzooxazol-2-y...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062257(2-({[(E)-5-Benzooxazol-2-yl-2-(4-chloro-phenyl)-1-...)
Affinity DataIC50:  28nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50404242(CHEMBL2114211)
Affinity DataIC50:  30nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062249(CHEMBL285434 | trisodium 5-[2-benzo[d][1,3]dioxol-...)
Affinity DataIC50:  45nMAssay Description:Inhibition of FTase in competitive manner with respect to FPP (farnesyl diphosphate) at 6.0 microM FPP and 0.36 microM Ras peptide.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50404243(CHEMBL2114212 | CHEMBL3350688)
Affinity DataIC50:  50nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062253(2-({[(E)-2-(4-Chloro-phenyl)-1-methyl-5-naphthalen...)
Affinity DataIC50:  51nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50223417(CHEMBL3350292)
Affinity DataIC50: >100nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062255(2-({[2,3-Bis-(4-chloro-phenyl)-1-methyl-propyl]-na...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50062254(2-({[2,3-Bis-(4-chloro-phenyl)-1-methyl-propyl]-me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Farnesyltransferase from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620495(3,5-Bis((4-borono-2-fluorobenzamido)methyl)benzoic...)
Affinity DataKd:  3.10E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620495(3,5-Bis((4-borono-2-fluorobenzamido)methyl)benzoic...)
Affinity DataKd:  8.60E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620496(3,5-Bis((4-borono-3-fluorobenzamido)methyl)benzoic...)
Affinity DataKd:  3.40E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620496(3,5-Bis((4-borono-3-fluorobenzamido)methyl)benzoic...)
Affinity DataKd:  5.40E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620497(N,N′-bis(4-borono-3-fluorobenzamido)-N-ethyl...)
Affinity DataKd:  2.70E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620497(N,N′-bis(4-borono-3-fluorobenzamido)-N-ethyl...)
Affinity DataKd:  1.60E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620498((S)-2,4-bis(4-borono-3-fluorobenzamido)butanoic ac...)
Affinity DataKd:  2.60E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620498((S)-2,4-bis(4-borono-3-fluorobenzamido)butanoic ac...)
Affinity DataKd:  6.50E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620499(N-(7-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  8.00E+5nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620499(N-(7-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  4.00E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620500(3,5-Bis((7-fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,...)
Affinity DataKd:  1.10E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620501(N-(5-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  1.50E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620501(N-(5-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  2.41E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620502(N-(4-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  2.70E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620502(N-(4-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  3.40E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620503(N-(6-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  2.60E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620503(N-(6-Fluoro-1-hydroxy-1,3-dihydrobenzo[c][1,2]oxab...)
Affinity DataKd:  6.79E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620504(N2,N6-Bis(6-fluoro-1-hydroxy-1,3-dihydrobenzo[c][1...)
Affinity DataKd:  3.20E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620504(N2,N6-Bis(6-fluoro-1-hydroxy-1,3-dihydrobenzo[c][1...)
Affinity DataKd:  3.52E+8nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620505(3-Borono-5-((3-borono-4-fluorophenyl)sulfonyl)-4-f...)
Affinity DataKd:  1.80E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620505(3-Borono-5-((3-borono-4-fluorophenyl)sulfonyl)-4-f...)
Affinity DataKd:  1.70E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620506(3-Borono-5-(3-borono-5-fluorobenzoyl)benzoic acid ...)
Affinity DataKd:  1.10E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620506(3-Borono-5-(3-borono-5-fluorobenzoyl)benzoic acid ...)
Affinity DataKd:  1.80E+7nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620507(3-Borono-5-(5-borono-2,4-difluorobenzoyl)benzoic a...)
Affinity DataKd:  3.00E+5nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

US Patent
LigandPNGBDBM620507(3-Borono-5-(5-borono-2,4-difluorobenzoyl)benzoic a...)
Affinity DataKd:  4.00E+6nMAssay Description:The alizarin-red binding assay is a colorimetric assay used to determine the inhibition affinity of boronate compounds to glucose. The assay is based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 104 total ) | Next | Last >>
Jump to: