TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to Trypanosoma brucei rhodesainMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of VEGFR2 by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:To characterize the type and extent inhibition of papain by fukugetin, papain (0.04 nM) was incubated with four concentrations of fukugetin (1.5, 3, ...More data for this Ligand-Target Pair
Affinity DataKi: 6.20E+3nMAssay Description:The iNOS activity assay was based on the method of hemoglobin assay previously described with slight modifications. The activity of the enzyme was de...More data for this Ligand-Target Pair
Affinity DataKi: 1.34E+4nMAssay Description:To characterize the type and extent inhibition of papain by fukugetin, papain (0.04 nM) was incubated with four concentrations of fukugetin (1.5, 3, ...More data for this Ligand-Target Pair
Affinity DataKi: 2.94E+4nMAssay Description:The iNOS activity assay was based on the method of hemoglobin assay previously described with slight modifications. The activity of the enzyme was de...More data for this Ligand-Target Pair
Affinity DataKi: 5.72E+4nMAssay Description:The iNOS activity assay was based on the method of hemoglobin assay previously described with slight modifications. The activity of the enzyme was de...More data for this Ligand-Target Pair
Affinity DataKi: 2.41E+5nMAssay Description:The iNOS activity assay was based on the method of hemoglobin assay previously described with slight modifications. The activity of the enzyme was de...More data for this Ligand-Target Pair
Affinity DataKi: 2.59E+5nMAssay Description:The iNOS activity assay was based on the method of hemoglobin assay previously described with slight modifications. The activity of the enzyme was de...More data for this Ligand-Target Pair
Affinity DataKi: 7.60E+5nMAssay Description:The iNOS activity assay was based on the method of hemoglobin assay previously described with slight modifications. The activity of the enzyme was de...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured for ...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured for ...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate by fluorimetric analysis relative to controlMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate by fluorimetric analysis relative to controlMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured for ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured for ...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition measured f...More data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate by fluorimetric analysis relative to controlMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate by fluorimetric analysis relative to controlMore data for this Ligand-Target Pair
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Federal University Of Alagoas
Curated by ChEMBL
Federal University Of Alagoas
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesain using Z-FR-AMC as substrate by fluorimetric analysis relative to controlMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 278nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 192nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 192nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 167nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 167nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 91nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 91nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Competitive inhibition of VEGFR2 by qPCR methodMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 278nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 286nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 286nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 222nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 384nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 384nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Instituto Tecnol£Gico E Nuclear
Curated by ChEMBL
Affinity DataKd: 222nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair