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Found 118 with Last Name = 'santra' and Initial = 's'
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50124566((R)-2-((R)-(2-ethoxyphenoxy)(phenyl)methyl)morphol...)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062762(CHEMBL3397792)
Affinity DataKi:  0.710nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062765(CHEMBL3397793)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50444862(CHEMBL3099493)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062769(CHEMBL3397803)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062752(CHEMBL3397805)
Affinity DataKi:  4.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062755(CHEMBL3397798)
Affinity DataKi:  5.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50444861(CHEMBL3099494)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062760(CHEMBL3397809)
Affinity DataKi:  7.40nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50444860(CHEMBL3099495)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062769(CHEMBL3397803)
Affinity DataKi:  8.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062764(CHEMBL3397800)
Affinity DataKi:  9nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062766(CHEMBL3397801)
Affinity DataKi:  9.30nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062753(CHEMBL3397806)
Affinity DataKi:  10nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataKi:  12.2nMAssay Description:Inhibition of SERT in rat cerebral cortex assessed as [3H]serotonin accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50343477((3S,6S)-6-Benzhydryl-N-(4-methoxybenzyl)tetrahydro...)
Affinity DataKi:  12.9nMAssay Description:Inhibition of SERT in rat cerebral cortex assessed as [3H]serotonin accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190608(CHEMBL213627 | cis-(3S,6S)-(6-benzhydryl-tetrahydr...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062761(CHEMBL3397810)
Affinity DataKi:  13nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062760(CHEMBL3397809)
Affinity DataKi:  13nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190609((2S,4R,5R)-5-(4-methoxybenzylamino)-2-benzhydryl-t...)
Affinity DataKi:  14.7nMAssay Description:Inhibition of SERT in rat cerebral cortex assessed as [3H]serotonin accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50343477((3S,6S)-6-Benzhydryl-N-(4-methoxybenzyl)tetrahydro...)
Affinity DataKi:  15.9nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataKi:  16.2nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062770(CHEMBL3397804)
Affinity DataKi:  17nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062759(CHEMBL3397808)
Affinity DataKi:  20nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190601((2S,4R,5R)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  25nMAssay Description:Inhibition of SERT in rat cerebral cortex assessed as [3H]serotonin accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062762(CHEMBL3397792)
Affinity DataKi:  25nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190601((2S,4R,5R)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062770(CHEMBL3397804)
Affinity DataKi:  26nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062752(CHEMBL3397805)
Affinity DataKi:  26nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062755(CHEMBL3397798)
Affinity DataKi:  27nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062768(CHEMBL3397802)
Affinity DataKi:  27nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062759(CHEMBL3397808)
Affinity DataKi:  28nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50343470((3S,6S)-6-Benzhydryl-N-(pyridin-4-ylmethyl)tetrahy...)
Affinity DataKi:  28.3nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062763(CHEMBL3397807)
Affinity DataKi:  29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062768(CHEMBL3397802)
Affinity DataKi:  29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062761(CHEMBL3397810)
Affinity DataKi:  29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(CHEMBL211077 | cis-(3S,6S)-(6-benzhydryl-tetrahydr...)
Affinity DataKi:  29.1nMAssay Description:Inhibition of SERT in rat cerebral cortex assessed as [3H]serotonin accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062757(CHEMBL3397795)
Affinity DataKi:  30nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(CHEMBL211077 | cis-(3S,6S)-(6-benzhydryl-tetrahydr...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50343473(3-((((3S,6S)-6-Benzhydryltetrahydro-2H-pyran-3-yl)...)
Affinity DataKi:  31.3nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062767(CHEMBL3397794)
Affinity DataKi:  34nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062765(CHEMBL3397793)
Affinity DataKi:  34nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062753(CHEMBL3397806)
Affinity DataKi:  37nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190609((2S,4R,5R)-5-(4-methoxybenzylamino)-2-benzhydryl-t...)
Affinity DataKi:  37.4nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062756(CHEMBL3397799)
Affinity DataKi:  38nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50444871(CHEMBL3099502)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-dopamine from rat cerebral cortex NET after 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50343473(3-((((3S,6S)-6-Benzhydryltetrahydro-2H-pyran-3-yl)...)
Affinity DataKi:  40.1nMAssay Description:Inhibition of SERT in rat cerebral cortex assessed as [3H]serotonin accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50343474((3S,6S)-6-Benzhydryl-N-(thiophen-2-ylmethyl)tetrah...)
Affinity DataKi:  41.4nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50062764(CHEMBL3397800)
Affinity DataKi:  42nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(CHEMBL211077 | cis-(3S,6S)-(6-benzhydryl-tetrahydr...)
Affinity DataKi:  42nMAssay Description:Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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