TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Mixed-type inhibition of electric eel AChE preincubated for 5 mins followed by varying levels acetylthiocholine iodide substrate addition by Lineweav...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Inhibition of human Protein kinase C beta 2More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 356nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 404nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 423nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 583nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 778nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
Affinity DataIC50: 5.49E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 5.76E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mazandaran
Curated by ChEMBL
University Of Mazandaran
Curated by ChEMBL
Affinity DataIC50: 6.22E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min...More data for this Ligand-Target Pair
Affinity DataIC50: 7.14E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 9.91E+3nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibitory activity against HepG2 Squalene Synthase (SQS)More data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 5.41E+4nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair
Affinity DataIC50: 7.43E+4nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured for 1 min by E...More data for this Ligand-Target Pair