TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 3.79E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 7.62E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataKi: 9.70E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 34.3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 85.4nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 89.7nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 114nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 165nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 174nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 177nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College Of Pharmaceutical Sciences
Curated by ChEMBL
University College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 191nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair