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Found 104 with Last Name = 'saunders' and Initial = 'l'
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50154337(6-((5S,11S,13aR)-5-benzyl-8,8-dimethyl-4,7,10,13-t...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50154337(6-((5S,11S,13aR)-5-benzyl-8,8-dimethyl-4,7,10,13-t...)
Affinity DataIC50:  21nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50154337(6-((5S,11S,13aR)-5-benzyl-8,8-dimethyl-4,7,10,13-t...)
Affinity DataIC50:  40nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375534(CHEMBL259517)
Affinity DataIC50:  130nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50:  240nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50274119(CHEMBL4126343)
Affinity DataIC50:  340nMAssay Description:Inhibition of Dengue virus 4 NS5 full length RdRp activity using RNA as template assessed as inhibition of NTPs incorporation after 90 mins by FAPA a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50274120(CHEMBL3417270)
Affinity DataIC50:  360nMAssay Description:Inhibition of Dengue virus 2 NS5 full length RdRp activity using RNA as template/primer assessed as inhibition of [alpha3P]GTP incorporation by SDS-P...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50115659((S)-3-biphenyl-4-yl-2-(7-hydroxycarbamoyl-heptanoy...)
Affinity DataIC50:  440nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375542(CHEMBL261492)
Affinity DataIC50:  570nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375540(CHEMBL259708)
Affinity DataIC50:  590nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375548(CHEMBL259434)
Affinity DataIC50:  630nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50274124(CHEMBL4125966 | US10793591, Compound 12)
Affinity DataIC50:  650nMAssay Description:Inhibition of Dengue virus RdRp activity using 5'-(TCAG)20(TCCAAG)14(TCAG)20-3' as template measured after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375534(CHEMBL259517)
Affinity DataIC50:  690nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50:  750nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant SIRT2 by fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant SIRT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375534(CHEMBL259517)
Affinity DataIC50:  960nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375535(CHEMBL264411)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50115659((S)-3-biphenyl-4-yl-2-(7-hydroxycarbamoyl-heptanoy...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant SIRT2 by radioactive deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375536(CHEMBL409526)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375548(CHEMBL259434)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50115659((S)-3-biphenyl-4-yl-2-(7-hydroxycarbamoyl-heptanoy...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50274121(CHEMBL4127092)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Dengue virus RdRp activity using 5'-(TCAG)20(TCCAAG)14(TCAG)20-3' as template measured after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375543(CHEMBL261272)
Affinity DataIC50:  1.68E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375546(CHEMBL406734)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375539(CHEMBL264926)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50274122(CHEMBL4127819)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Dengue virus RdRp activity using 5'-(TCAG)20(TCCAAG)14(TCAG)20-3' as template measured after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375545(CHEMBL260080)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375543(CHEMBL261272)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375537(CHEMBL261587)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375537(CHEMBL261587)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50199961(3-(1-{2-[1-(1,4-dioxa-spiro[4.5]dec-2-yl)-3-hydrox...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human recombinant SIRT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375541(CHEMBL409860)
Affinity DataIC50:  2.55E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375538(CHEMBL427776)
Affinity DataIC50:  2.61E+3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Novartis Institute For Tropical Diseases

Curated by ChEMBL
LigandPNGBDBM50274125(CHEMBL4127565)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of Dengue virus RdRp activity using 5'-(TCAG)20(TCCAAG)14(TCAG)20-3' as template measured after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50199962(3-(1-{2-[1-(1,4-dioxa-spiro[4.5]dec-2-yl)-3-hydrox...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human recombinant SIRT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375544(CHEMBL263884)
Affinity DataIC50:  2.85E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50:  2.96E+3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375548(CHEMBL259434)
Affinity DataIC50:  2.98E+3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375539(CHEMBL264926)
Affinity DataIC50:  3.01E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375535(CHEMBL264411)
Affinity DataIC50:  3.03E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375536(CHEMBL409526)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Rattus norvegicus)
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375546(CHEMBL406734)
Affinity DataIC50:  3.19E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375540(CHEMBL259708)
Affinity DataIC50:  3.34E+3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human SIRT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human SIRT1 by fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375540(CHEMBL259708)
Affinity DataIC50:  4.02E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375541(CHEMBL409860)
Affinity DataIC50:  4.09E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50375538(CHEMBL427776)
Affinity DataIC50:  4.49E+3nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in human 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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