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Found 7 with Last Name = 'sawkar' and Initial = 'a'
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
TBA

Curated by ChEMBL
LigandPNGBDBM50108799((2-[N -(2-hydroxyethyl)]-N -(4-methoxybenzenesulfo...)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of Myosin Light Chain kinase (MLCK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM18370(N-(adamantan-1-yl)-5-[(3R,4R,5R)-3,4-dihydroxy-5-(...)
Affinity DataIC50:  1.10E+4nMpH: 5.0 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 365 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM18369(N-(adamantan-1-yl)-4-[(3R,4R,5R)-3,4-dihydroxy-5-(...)
Affinity DataIC50:  1.80E+4nMpH: 5.0 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 365 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM18371(N-(adamantan-1-yl)-6-[(3R,4R,5R)-3,4-dihydroxy-5-(...)
Affinity DataIC50:  9.40E+4nMpH: 5.0 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 365 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
TBA

Curated by ChEMBL
LigandPNGBDBM50108800(11-(3-Imino-5,6-dihydro-3H-benzo[h]cinnolin-2-yl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Myosin Light Chain kinase (MLCK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM18368(2,5-anhydro-2,5-imino-D-glucitol based compound, 2...)
Affinity DataIC50:  3.93E+5nMpH: 5.0 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 365 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM18367(2,5-anhydro-2,5-imino-D-glucitol based compound, 1...)
Affinity DataIC50:  5.07E+5nMpH: 5.0 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 365 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed