Compile Data Set for Download or QSAR
maximum 50k data
Found 23 with Last Name = 'scarf' and Initial = 'am'
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50350912(CHEMBL1817978)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50185957(CHEMBL205767 | N-(2-isopropoxybenzyl)-N-(4-chloro-...)
Affinity DataKi:  0.920nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50350912(CHEMBL1817978)
Affinity DataKi:  1.19nMAssay Description:Displacement of [3H]PK11195 from TSPO in human HEK293 mitochondrial fractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenateMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50253713(CHEMBL461828 | N-benzyl-2-(5-chloro-2-(4-chlorophe...)
Affinity DataKi:  3.33nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50350912(CHEMBL1817978)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial fractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50045877(2-(2-(4-fluorophenyl)-1H-indol-3-yl)-N,N-dihexylac...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  7.11nMAssay Description:Displacement of [3H]PK11195 from TSPO in human HEK293 mitochondrial fractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  8.20nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial fractionMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  28nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  144nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  398nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  806nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Cea

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKd:  0.600nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat cortexMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM50255226((7-chloro-N,N,5-trimethyl-4-oxo-3-phenyl-3,5-dihyd...)
Affinity DataKd:  3nMAssay Description:Displacement of [3H]SSR180575 from TSPO in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Cea

Curated by ChEMBL
LigandPNGBDBM22040(4 -chlorodiazepam | 4' Cl-diazepam | 7-chloro-...)
Affinity DataKd:  1.10nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kainate lesioned striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed