TargetPOU domain, class 2, transcription factor 1(Homo sapiens (Human))
Nippon Boehringer Ingelheim
Curated by ChEMBL
Nippon Boehringer Ingelheim
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of OCT1 (unknown origin) expressed in HEK293 cells assessed as reduction of [14C]metformin substrate uptake at 100 uM by liquid scintillat...More data for this Ligand-Target Pair
TargetPOU domain, class 2, transcription factor 1(Homo sapiens (Human))
Nippon Boehringer Ingelheim
Curated by ChEMBL
Nippon Boehringer Ingelheim
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of OCT1 (unknown origin) expressed in HEK293 cells assessed as reduction of [ethyl 1-14C]TEA substrate uptake at 100 uM by liquid scintill...More data for this Ligand-Target Pair
TargetPOU domain, class 2, transcription factor 2(Homo sapiens (Human))
Nippon Boehringer Ingelheim
Curated by ChEMBL
Nippon Boehringer Ingelheim
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of OCT2 (unknown origin) expressed in HEK293 cells assessed as reduction of [14C]metformin substrate uptake at 100 uM by liquid scintillat...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Nippon Boehringer Ingelheim
Curated by ChEMBL
Nippon Boehringer Ingelheim
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction of [3H]E-sul substrate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Nippon Boehringer Ingelheim
Curated by ChEMBL
Nippon Boehringer Ingelheim
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction of [3H]E217betaG substrate uptake by liquid scintillation coun...More data for this Ligand-Target Pair