Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.60E+3nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 120nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 170nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 170nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]iodotyrosyl from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 210nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 214nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 230nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 240nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 240nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 247nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 260nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 280nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 290nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 420nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Displacement of [125I]iodotyrosyl from human SST4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Displacement of [I125I]MCH from human MCH1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 470nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 490nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Displacement of [125I]iodotyrosyl from human SST3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetIsoform Tau-F of Microtubule-associated protein tau(Homo sapiens (Human))
The Ohio State University
The Ohio State University
Affinity DataIC50: 520nMpH: 7.4Assay Description:The Tau content of fractions was determined by dot blot analysis using nitrocellulose membranes (0.2 μm porosity) as described previously [Cisek...More data for this Ligand-Target Pair