BindingDB PrimarySearch_ki

Found 64 with Last Name = 'scheepstra' and Initial = 'm'

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50106301(CHEMBL3598140)

IC50: 7.80nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50106301(CHEMBL3598140)

IC50: 7.80nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50106301(CHEMBL3598140)

IC50: 9.40nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50106301(CHEMBL3598140)

IC50: 13nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50106301(CHEMBL3598140)

IC50: 17nMAssay Description:Displacement of Alexa647-labeled MRL-87 from human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519883(CHEMBL4522217)

IC50: 94nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519883(CHEMBL4522217)

IC50: 118nMAssay Description:Displacement of Alexa647-labeled MRL-87 from human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3...More data for this Ligand-Target Pair

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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519883(CHEMBL4522217)

IC50: 138nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519881(CHEMBL4435145)

IC50: 180nMAssay Description:Displacement of Alexa647-labeled MRL-87 from human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519883(CHEMBL4522217)

IC50: 248nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519883(CHEMBL4522217)

IC50: 264nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519881(CHEMBL4435145)

IC50: 269nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519881(CHEMBL4435145)

IC50: 300nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519881(CHEMBL4435145)

IC50: 425nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519881(CHEMBL4435145)

IC50: 547nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519885(CHEMBL4469931)

IC50: 1.09E+3nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519884(CHEMBL4438380)

IC50: 1.75E+3nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519882(CHEMBL4465726)

IC50: 6.62E+3nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)

IC50: 7.01E+3nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

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3D Structure (crystal)

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50106301(CHEMBL3598140)

IC50: 7.20E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519891(CHEMBL4452679)

IC50: 8.76E+3nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519878(CHEMBL4550831)

IC50: 9.60E+3nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519881(CHEMBL4435145)

IC50: 1.47E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519886(CHEMBL4587804)

IC50: 3.09E+4nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)

IC50: 3.36E+4nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519880(CHEMBL4518713)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519894(CHEMBL4436630)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519893(CHEMBL4437814)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519890(CHEMBL4452409)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519895(CHEMBL4435027)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519886(CHEMBL4587804)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519887(CHEMBL4457177)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519891(CHEMBL4452679)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519879(CHEMBL4574983)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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KEGG PC cid PC sid

Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519889(CHEMBL4466846)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519888(CHEMBL4444484)

IC50: >5.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519888(CHEMBL4444484)

IC50: 5.35E+4nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519893(CHEMBL4437814)

IC50: 6.26E+4nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519890(CHEMBL4452409)

IC50: 7.39E+4nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519878(CHEMBL4550831)

IC50: 7.86E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)

IC50: 8.54E+4nMAssay Description:Competitive inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) ass...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519894(CHEMBL4436630)

IC50: 9.11E+4nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519883(CHEMBL4522217)

IC50: 9.93E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519882(CHEMBL4465726)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519884(CHEMBL4438380)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519885(CHEMBL4469931)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Peroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519892(CHEMBL4514441)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-act...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519892(CHEMBL4514441)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519889(CHEMBL4466846)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL

PNG

BDBM50519887(CHEMBL4457177)

IC50: >1.00E+5nMAssay Description:Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inh...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

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