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Found 89 with Last Name = 'schiaffella' and Initial = 'f'
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086666(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4-{3-[4-(2...)
Affinity DataKi:  1.30nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040072(4-Chloro-benzene-1,3-disulfonic acid 3-amide 1-({2...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040065(5-[3-(tert-butylamino)-2-hydroxypropoxy]-3,4-dihyd...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086666(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4-{3-[4-(2...)
Affinity DataKi:  2.70nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040076(4-Chloro-benzene-1,3-disulfonic acid 3-amide 1-({2...)
Affinity DataKi:  5.20nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086666(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4-{3-[4-(2...)
Affinity DataKi:  5.30nMAssay Description:Compound was evaluated for its Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat hea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040073(4-Chloro-N-{2-[2-hydroxy-3-(3-oxo-3,4-dihydro-2H-b...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040069(2-Chloro-5-{2-[2-hydroxy-3-(3-oxo-3,4-dihydro-2H-b...)
Affinity DataKi:  7.80nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086668(7-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  8.30nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50218566(CHEMBL140477)
Affinity DataKi:  14nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040074(2-Chloro-5-{2-[2-hydroxy-3-(naphthalen-1-yloxy)-pr...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50218562(CHEMBL141194)
Affinity DataKi:  15nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086677(6-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  16nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086673(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4H-benzo[1...)
Affinity DataKi:  20nMAssay Description:Compound was evaluated for its Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat hea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086665(7-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi:  20nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50218563(CHEMBL341723)
Affinity DataKi:  23nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086673(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4H-benzo[1...)
Affinity DataKi:  23nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50218565(CHEMBL143288)
Affinity DataKi:  23nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040070(8-tert-Butylamino-2-(3-hydroxy-propoxy)-4H-benzo[1...)
Affinity DataKi:  24nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086670(8-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  27nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040071(2-Chloro-5-{4-[2-hydroxy-3-(naphthalen-1-yloxy)-pr...)
Affinity DataKi:  31nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218563(CHEMBL341723)
Affinity DataKi:  32nMAssay Description:Alpha-2 adrenergic receptor binding affinity by measuring the displacement of [3H]clonidine binding in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086662(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi:  38nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...)
Affinity DataKi:  39nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086679(8-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi:  60nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50218567(CHEMBL142859)
Affinity DataKi:  73nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086670(8-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  88nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086663(6-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi:  90nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218566(CHEMBL140477)
Affinity DataKi:  99nMAssay Description:Alpha-2 adrenergic receptor binding affinity by measuring the displacement of [3H]clonidine binding in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50086660(6-{3-[4-(4-Fluoro-benzoyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi:  100nMAssay Description:Alpha-2 adrenergic receptor binding affinity by measuring the displacement of [3H]clonidine binding in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040066(2-Chloro-5-{4-[2-hydroxy-3-(3-oxo-3,4-dihydro-2H-b...)
Affinity DataKi:  140nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040068(4-Chloro-benzene-1,3-disulfonic acid 3-amide 1-({2...)
Affinity DataKi:  160nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040075(4-Chloro-N-{2-[2-hydroxy-3-(2-oxo-1,2,3,4-tetrahyd...)
Affinity DataKi:  300nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086670(8-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  330nMAssay Description:Compound was evaluated for its Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat hea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218562(CHEMBL141194)
Affinity DataKi:  370nMAssay Description:Alpha-2 adrenergic receptor binding affinity by measuring the displacement of [3H]clonidine binding in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50086662(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi:  440nMAssay Description:Alpha-2 adrenergic receptor binding affinity by measuring the displacement of [3H]clonidine binding in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50086666(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4-{3-[4-(2...)
Affinity DataKi:  530nMAssay Description:Alpha-2 adrenergic receptor binding affinity by measuring the displacement of [3H]clonidine binding in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50218564(CHEMBL143923)
Affinity DataKi:  540nMAssay Description:Alpha-1 adrenergic receptor binding affinity by measuring the displacement of [3H]prazosin binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040067(4-Chloro-N-{2-[2-hydroxy-3-(naphthalen-1-yloxy)-pr...)
Affinity DataKi:  820nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086675(8-{3-[4-(4-Fluoro-benzoyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086664(8-{3-[4-(Furan-2-carbonyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086672(7-{3-[4-(Furan-2-carbonyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086660(6-{3-[4-(4-Fluoro-benzoyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...)
Affinity DataKi:  1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086663(6-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat heart ; Not Active means Ki >1000 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086664(8-{3-[4-(Furan-2-carbonyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat heart ; Not Active means Ki >1000 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086668(7-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Università

Curated by ChEMBL
LigandPNGBDBM50086662(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]-DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50086665(7-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat heart ; Not Active means Ki >1000 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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