Affinity DataIC50: 140nMAssay Description:Inhibition of biotinylated polymeric fucose binding to Pseudomonas aeruginosa LecB expressed in Escherichia coli BL21(DE3) preincubated for 1 hr foll...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PA14 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PA14 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PAO1 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PAO1 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of COX1 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as reduction in ethidium bromide efflux by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of COX2 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of COX2 in human whole blood after 15 minsMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of COX2 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of COX2 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of COX1 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as reduction in ethidium bromide efflux by fluorescence assayMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of COX1 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of COX1 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of COX2 in human whole blood after 15 minsMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as reduction in ethidium bromide efflux by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of COX1 in human whole blood after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa LecBMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX2 in human whole blood after 15 minsMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX1 in human whole blood after 15 minsMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtA using dabcyl-QALPETGEE-edans as substrate preincubated for 1 hr followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.92E+5nMAssay Description:Inhibition of Staphylococcus aureus SrtAMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 2.09E+5nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair
TargetDehydrogenase/reductase SDR family member 9(Rattus norvegicus)
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 2.09E+5nMAssay Description:Inhibition of rat liver 3-alpha-HSD assessed as 5-beta-dihydrocortisone reductionMore data for this Ligand-Target Pair