Compile Data Set for Download or QSAR
maximum 50k data
Found 17 with Last Name = 'schlosburg' and Initial = 'j'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360023(CHEMBL1928337)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360023(CHEMBL1928337)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataKi:  7.80E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant FAAH expressed in Cos7 cells after 30 mins by using anandamide as a substrate by LC-MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant MAGL expressed in Cos7 cells after 30 mins by using 2-AG as a substrate by LC-MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  8nMAssay Description:Inhibition of MAGL in C57B1/6J mouse brain membrane after 30 mins by using 2-AG as a substrate by LC-MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of FAAH in C57B1/6J mouse brain membrane after 20 mins by using oleamide as a substrate by LC-MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360021(CHEMBL1164701)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50128581(Biphenyl-3-yl-carbamic acid cyclohexyl ester | CHE...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of MAGL in Wistar rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360021(CHEMBL1164701)
Affinity DataIC50:  3.07E+5nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM85515(Ampyrone | CAS_83-07-8 | EN300-17058 | NSC_2151 | ...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM85515(Ampyrone | CAS_83-07-8 | EN300-17058 | NSC_2151 | ...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50054471((5Z,8Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed