Affinity DataIC50: 0.0320nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]-ET-1 binding to rat aorta membrane Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Inhibition of [125I]-ET-1 binding to rat aorta membrane Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:In vitro inhibition of human renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Compound was tested in vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:The compound was tested in vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:In vitro inhibition of human renin.More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMpH: 5.5Assay Description:In vitro inhibitory activity against human plasma renin at pH 5.5 for suppression of angiotensin I formation.More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:In vitro inhibition of human renin.More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Ability to displace [125I]-Endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:In vitro inhibition of human renin.More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:In vitro inhibition of human renin.More data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:In vitro inhibition of human renin.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMpH: 5.5Assay Description:In vitro inhibitory activity against human plasma renin at pH 5.5 for suppression of angiotensin I formation.More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Compound was tested in vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:In vitro for inhibitory activity against human reninMore data for this Ligand-Target Pair