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Found 121 with Last Name = 'schneck' and Initial = 'j'
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417996(CHEMBL1672434)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418002(CHEMBL1672427)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417991(CHEMBL1672425)
Affinity DataIC50:  7.94nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417991(CHEMBL1672425)
Affinity DataIC50:  7.94nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31647(tetrahydrobenzothiophene (THBT), 21)
Affinity DataIC50:  10nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417998(CHEMBL1672426)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31648(tetrahydrobenzothiophene (THBT), 22)
Affinity DataIC50:  25nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418002(CHEMBL1672427)
Affinity DataIC50:  25.1nMAssay Description:Inhibition of human recombinant cathepsin L after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418001(CHEMBL1672421 | US11414402, Example 6)
Affinity DataIC50:  31.6nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417991(CHEMBL1672425)
Affinity DataIC50:  39.8nMAssay Description:Inhibition of human recombinant cathepsin L after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417996(CHEMBL1672434)
Affinity DataIC50:  39.8nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31644(tetrahydrobenzothiophene (THBT), 23)
Affinity DataIC50:  50nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31637(tetrahydrobenzothiophene (THBT), 6)
Affinity DataIC50:  50nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417997(CHEMBL1672423)
Affinity DataIC50:  63.1nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31638(tetrahydrobenzothiophene (THBT), 13a)
Affinity DataIC50:  79nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417998(CHEMBL1672426)
Affinity DataIC50:  79.4nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31649(tetrahydrobenzothiophene (THBT), 24)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417995(CHEMBL1672433)
Affinity DataIC50:  126nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418002(CHEMBL1672427)
Affinity DataIC50:  126nMAssay Description:Inhibition of human recombinant cathepsin S after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31648(tetrahydrobenzothiophene (THBT), 22)
Affinity DataIC50:  126nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31647(tetrahydrobenzothiophene (THBT), 21)
Affinity DataIC50:  126nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418000(CHEMBL1672432)
Affinity DataIC50:  158nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417989(CHEMBL1672422 | US11414402, Example 7)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31636(tetrahydrobenzothiophene (THBT), 4)
Affinity DataIC50:  200nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418000(CHEMBL1672432)
Affinity DataIC50:  251nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31636(tetrahydrobenzothiophene (THBT), 4)
Affinity DataIC50:  316nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417989(CHEMBL1672422 | US11414402, Example 7)
Affinity DataIC50:  316nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417991(CHEMBL1672425)
Affinity DataIC50:  316nMAssay Description:Inhibition of human recombinant cathepsin S after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418001(CHEMBL1672421 | US11414402, Example 6)
Affinity DataIC50:  316nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31644(tetrahydrobenzothiophene (THBT), 23)
Affinity DataIC50:  398nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31650(tetrahydrobenzothiophene (THBT), 25)
Affinity DataIC50:  398nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31637(tetrahydrobenzothiophene (THBT), 6)
Affinity DataIC50:  501nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417996(CHEMBL1672434)
Affinity DataIC50:  501nMAssay Description:Inhibition of human recombinant cathepsin L after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418001(CHEMBL1672421 | US11414402, Example 6)
Affinity DataIC50:  501nMAssay Description:Inhibition of human recombinant cathepsin S after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417995(CHEMBL1672433)
Affinity DataIC50:  631nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418003(CHEMBL1672419)
Affinity DataIC50:  631nMAssay Description:Inhibition of human recombinant cathepsin L after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31640(tetrahydrobenzothiophene (THBT), 14)
Affinity DataIC50:  631nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417990(CHEMBL1672424)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant cathepsin C after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50514671(CHEMBL4532803)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of full length C-terminal His6-tagged ERAP1 (unknown origin)-mediated antigenic epitope destruction assessed as inhibition of trimming of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50514671(CHEMBL4532803)
Affinity DataIC50:  1.00E+3nMAssay Description:Activation of full length C-terminal His6-tagged ERAP1 (unknown origin)-mediated fluorogenic Leu-AMC substrate hydrolysis after 60 mins by Rapidfire-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417993(CHEMBL1672430)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417996(CHEMBL1672434)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant cathepsin S after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417990(CHEMBL1672424)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human recombinant cathepsin L after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417998(CHEMBL1672426)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human recombinant cathepsin L after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417990(CHEMBL1672424)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human recombinant cathepsin B after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418003(CHEMBL1672419)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human recombinant cathepsin K after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31646(tetrahydrobenzothiophene (THBT), 20)
Affinity DataIC50:  1.26E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50514671(CHEMBL4532803)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of full length C-terminal His6-tagged ERAP1 (unknown origin)-mediated chicken ovalbumin antigenic epitope processing assessed as reduction...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM31642(tetrahydrobenzothiophene (THBT), 16)
Affinity DataIC50:  1.26E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50418003(CHEMBL1672419)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of human recombinant cathepsin S after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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