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Found 89 with Last Name = 'schoen' and Initial = 'wr'
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  10nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  12nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  16nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  16nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  18nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  20nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  25nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121048(2-[3-Butyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  28nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  30nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  40nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  65nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  110nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  110nMAssay Description:Binding affinity of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50:  120nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109332(1-[4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyr...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109338(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-py...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50:  190nMAssay Description:Binding affinity of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50:  190nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  190nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109319(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109316(1-[4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyr...)
Affinity DataIC50:  240nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109337(1-[5-Butyl-4-(4-fluoro-phenyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109339(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-py...)
Affinity DataIC50:  300nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109329(CHEMBL143664 | [4-(4-Fluoro-phenyl)-5-hexyl-2,6-di...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109323(CHEMBL140514 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331(CHEMBL24616 | [4-(4-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  400nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112484(2-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridi...)
Affinity DataIC50:  500nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109341(CHEMBL140268 | [4-(4-Fluoro-phenyl)-5-heptyl-2,6-d...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331(CHEMBL24616 | [4-(4-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  700nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331(CHEMBL24616 | [4-(4-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109318(CHEMBL143698 | [5-Butyl-4-(4-fluoro-phenyl)-2,6-di...)
Affinity DataIC50:  750nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112475(CHEMBL286098 | [4-(4-Chloro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  800nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112479((2,6-Diisopropyl-5-pentyl-4-p-tolyl-pyridin-3-yl)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109327(CHEMBL143609 | [5-Ethyl-4-(4-fluoro-phenyl)-2,6-di...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109325(CHEMBL140586 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121048(2-[3-Butyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112478(CHEMBL286555 | [4-(3,4-Difluoro-phenyl)-2,6-diisop...)
Affinity DataIC50:  1.10E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109336((2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-m...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109336((2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-m...)
Affinity DataIC50:  1.40E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109317((5-Ethyl-2,6-diisopropyl-4-phenyl-pyridin-3-yl)-me...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109315(CHEMBL140636 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322(CHEMBL114761 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration of the compound against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112485(CHEMBL277627 | [4-(2-Amino-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  2.30E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112483(CHEMBL25137 | [4-(3-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022578(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-nona...)
Affinity DataIC50:  4.00E+3nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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