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Found 109 with Last Name = 'schulz' and Initial = 'b'
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244756(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-1,2-benzisothi...)
Affinity DataKi:  28nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244756(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-1,2-benzisothi...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  800nMAssay Description:Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244751(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-4,5,6,7-tetrah...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244756(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-1,2-benzisothi...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of wild type MET assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of recombinant AXL assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of recombinant IGF1-R assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of recombinant PLK1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt-activated lipase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244756(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-1,2-benzisothi...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of cholesterol esterase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of recombinant SRC assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of recombinant FAK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of recombinant ARK5 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244753(5-Methyl-4-phenyl-2-(2,3,5,6-tetrafluoropyridin-4-...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of recombinant ARK5 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  3.33E+4nMAssay Description:Inhibition of recombinant IGF1-R assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of recombinant SRC assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  4.13E+4nMAssay Description:Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  4.53E+4nMAssay Description:Inhibition of recombinant PRK1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  5.49E+4nMAssay Description:Inhibition of recombinant PRK1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek6(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  6.78E+4nMAssay Description:Inhibition of recombinant NEK6 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  7.57E+4nMAssay Description:Inhibition of recombinant PLK1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  8.39E+4nMAssay Description:Inhibition of recombinant NEK2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244755(2-(Pyridin-4-yl)-4,5,6,7-tetrahydro-1,2-benzisothi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244703(2-(6-Chloropyridin-2-yl)-4,5,6,7-tetrahydro-1,2-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244703(2-(6-Chloropyridin-2-yl)-4,5,6,7-tetrahydro-1,2-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244703(2-(6-Chloropyridin-2-yl)-4,5,6,7-tetrahydro-1,2-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244703(2-(6-Chloropyridin-2-yl)-4,5,6,7-tetrahydro-1,2-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244703(2-(6-Chloropyridin-2-yl)-4,5,6,7-tetrahydro-1,2-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of acetylcholinesterase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt-activated lipase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244703(2-(6-Chloropyridin-2-yl)-4,5,6,7-tetrahydro-1,2-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of cholesterol esterase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244754(2-(2,3,4,5,6-Pentafluorophenyl)-4,5,6,7-tetrahydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244752(4,5-Dimethyl-2-(2,3,5,6-tetrafluoropyridin-4-yl)-i...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244705(2-(3,5-Difluoropyridin-2-yl)-4,5,6,7-tetrahydro-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244704(2-(6-Bromopyridin-2-yl)-4,5,6,7-tetrahydro-1,2-ben...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244755(2-(Pyridin-4-yl)-4,5,6,7-tetrahydro-1,2-benzisothi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244754(2-(2,3,4,5,6-Pentafluorophenyl)-4,5,6,7-tetrahydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244753(5-Methyl-4-phenyl-2-(2,3,5,6-tetrafluoropyridin-4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244752(4,5-Dimethyl-2-(2,3,5,6-tetrafluoropyridin-4-yl)-i...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244751(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-4,5,6,7-tetrah...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244705(2-(3,5-Difluoropyridin-2-yl)-4,5,6,7-tetrahydro-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244704(2-(6-Bromopyridin-2-yl)-4,5,6,7-tetrahydro-1,2-ben...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244756(2-(2,3,5,6-Tetrafluoropyridin-4-yl)-1,2-benzisothi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244755(2-(Pyridin-4-yl)-4,5,6,7-tetrahydro-1,2-benzisothi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of Leipzig

Curated by ChEMBL
LigandPNGBDBM50244754(2-(2,3,4,5,6-Pentafluorophenyl)-4,5,6,7-tetrahydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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