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Found 65 with Last Name = 'schulz' and Initial = 'f'
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314131((S,E)-Ethyl 4-((R)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  140nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314126((S)-Benzyl-2-[(Z)-3-((S)-1-benzyloxycarbonyl-2-phe...)
Affinity DataKi:  150nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using low concentration of enzyme by standard fluorescence assay in presence of de...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314130((S)-2-[(E)-3-((S)-1-Benzyloxycarbonyl-2-phenylethy...)
Affinity DataKi:  340nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using high concentration of enzyme by standard fluorescence assay in presence of d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  470nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  640nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using low concentration of enzyme by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  640nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using high concentration of enzyme by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314127((S)-Benzyl-2-{(Z)-3-[(S)-1-((S)-1-benzyloxycarbony...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314128((S,E)-Methyl 2-(4-Ethoxy-4-oxobut-2-enamido)-5-oxo...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314124((S,E)-ethyl 4-(tert-butoxycarbonylamino)-7-oxo-7-(...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assay in presence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314124((S,E)-ethyl 4-(tert-butoxycarbonylamino)-7-oxo-7-(...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50175214((2R,3R)-diethyl 1-((2S)-3-(azetidin-1-yl)-2-(tert-...)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibitory activity against cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314132((2S,5S,8S,11S,E)-1-Benzyl 16-ethyl 11-(3-amino-3-o...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50175213((2S,3S)-dibenzyl 1-((S)-2-(tert-butoxycarbonyl)-2-...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibitory activity against cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50314129((S,E)-3-((S)-1-Benzyloxycarbonyl-2-phenylethylcarb...)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346543(CHEMBL1797750)
Affinity DataIC50:  98nMAssay Description:Inhibition of SIRT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346550(CHEMBL270110)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of SIRT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged Sirt1 expressed in Escherichia coli using ZMAL as substrate after 4 hrs by homogeneous fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM3175(3-[1-[3-(Amidinothio)propyl]-3-indolyl]-4-(1-methy...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human C-terminally His6-tagged Sirt3 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346546(CHEMBL1797926)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346546(CHEMBL1797926)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged Sirt1 expressed in Escherichia coli using ZMAL as substrate after 4 hrs by homogeneous fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM74978(1,3-dihydrobenzo[e]benzimidazole-2-thione | CHEMBL...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged Sirt1 expressed in Escherichia coli using ZMAL as substrate after 4 hrs by homogeneous fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM74978(1,3-dihydrobenzo[e]benzimidazole-2-thione | CHEMBL...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521373(CHEMBL4573866)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of fluorescent labelled LBS3 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346547(CHEMBL1797919)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521373(CHEMBL4573866)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346545(CHEMBL1797923)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521372(CHEMBL4468809)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of fluorescent labelled LBS3 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521373(CHEMBL4573866)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of fluorescent labelled LBS1 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521369(CHEMBL4439456)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of fluorescent labelled LBS1 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346545(CHEMBL1797923)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged Sirt1 expressed in Escherichia coli using ZMAL as substrate after 4 hrs by homogeneous fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521370(CHEMBL4468972)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of fluorescent labelled LBS1 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521372(CHEMBL4468809)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of fluorescent labelled LBS1 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521372(CHEMBL4468809)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of fluorescent labelled LBS3 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521370(CHEMBL4468972)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of fluorescent labelled LBS3 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346548(CHEMBL1797922)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521382(CHEMBL4548393)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521370(CHEMBL4468972)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346544(CHEMBL1797920)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged Sirt1 expressed in Escherichia coli using ZMAL as substrate after 4 hrs by homogeneous fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50328901(4-(4-(Aminomethyl)-1H-1,2,3-triazol-1-yl)benzoic a...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346549(CHEMBL1797925)
Affinity DataIC50:  3.44E+4nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ernst-Moritz-Arndt University Greifswald

Curated by ChEMBL
LigandPNGBDBM50346544(CHEMBL1797920)
Affinity DataIC50:  3.83E+4nMAssay Description:Inhibition of human N-terminally His6-tagged Sirt2 using ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521381(CHEMBL4436463)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of fluorescent labelled LBS3 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521379(CHEMBL4449651)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521383(CHEMBL4559370)
Affinity DataIC50:  7.90E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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