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Found 3234 with Last Name = 'schulz-gasch' and Initial = 't'
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429823(CHEMBL2338173)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Hamburg

Curated by ChEMBL
LigandPNGBDBM50085406((2R,3R)-3-[(Biphenyl-4-carbonyl)-amino]-2-(3-carba...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429823(CHEMBL2338173)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein, adipocyte(Homo sapiens (Human))TBA
LigandPNGBDBM50197092(CHEMBL3947458)
Affinity DataKi:  12nMAssay Description:Inhibition of FABP4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Hamburg

Curated by ChEMBL
LigandPNGBDBM50114532((R)-2-{[(Biphenyl-4-carbonyl)-amino]-methyl}-3-(3-...)
Affinity DataKi:  20nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein, adipocyte(Homo sapiens (Human))TBA
LigandPNGBDBM50197094(CHEMBL3941588)
Affinity DataKi:  22nMAssay Description:Inhibition of FABP4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Homo sapiens (Human))TBA
LigandPNGBDBM50613583(CHEMBL5287034)
Affinity DataKi:  30nMAssay Description:Inhibition of FABP4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFatty acid-binding protein, heart(Homo sapiens (Human))TBA
LigandPNGBDBM50197091(CHEMBL1738980)
Affinity DataKi:  90nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, adipocyte(Homo sapiens (Human))TBA
LigandPNGBDBM50197091(CHEMBL1738980)
Affinity DataKi:  100nMAssay Description:Inhibition of FABP4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetFatty acid-binding protein, heart(Homo sapiens (Human))TBA
LigandPNGBDBM50613583(CHEMBL5287034)
Affinity DataKi:  150nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429830(CHEMBL2338182)
Affinity DataKi:  170nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429829(CHEMBL2338183)
Affinity DataKi:  200nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429826(CHEMBL2338186)
Affinity DataKi:  270nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429824(CHEMBL2338188)
Affinity DataKi:  320nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataKi:  350nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein, heart(Homo sapiens (Human))TBA
LigandPNGBDBM50197092(CHEMBL3947458)
Affinity DataKi:  380nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429826(CHEMBL2338186)
Affinity DataKi:  400nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429833(CHEMBL2338178)
Affinity DataKi:  460nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50197094(CHEMBL3941588)
Affinity DataKi:  490nMAssay Description:Inhibition of FABP5 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429831(CHEMBL2338181)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429832(CHEMBL2338179)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429825(CHEMBL2338187)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429827(CHEMBL2338185)
Affinity DataKi:  600nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429837(CHEMBL2338174)
Affinity DataKi:  770nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataKi:  790nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429832(CHEMBL2338179)
Affinity DataKi:  900nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429836(CHEMBL2338175)
Affinity DataKi:  990nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50197092(CHEMBL3947458)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of FABP5 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429830(CHEMBL2338182)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429824(CHEMBL2338188)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429829(CHEMBL2338183)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429828(CHEMBL2338184)
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429828(CHEMBL2338184)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429831(CHEMBL2338181)
Affinity DataKi:  4.90E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429837(CHEMBL2338174)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50613583(CHEMBL5287034)
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of FABP5 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429833(CHEMBL2338178)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429827(CHEMBL2338185)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429825(CHEMBL2338187)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429836(CHEMBL2338175)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein, heart(Homo sapiens (Human))TBA
LigandPNGBDBM50197094(CHEMBL3941588)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty acid-binding protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50197091(CHEMBL1738980)
Affinity DataKi: >2.30E+4nMAssay Description:Inhibition of FABP5 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50397965(CHEMBL2180789)
Affinity DataIC50:  0.0190nMAssay Description:Inhibition of full-length recombinant human PDE10A by scintillation proximity assayMore data for this Ligand-Target Pair
LigandPNGBDBM50613581(CHEMBL5286395)
Affinity DataIC50:  0.0630nMAssay Description:Inhibition of full-length recombinant human PDE10A by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50613582(CHEMBL5288570)
Affinity DataIC50:  0.102nMAssay Description:Inhibition of full-length recombinant human PDE10A by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCathepsin S(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM122478(US8729061, 8)
Affinity DataIC50:  0.296nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In DepthDetails US Patent
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