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Found 1071 with Last Name = 'schwarz' and Initial = 'm'
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50326722((Z)-3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoi...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50326722((Z)-3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoi...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410618(CHEMBL2113181)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410616(CHEMBL2113185)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM244799(US9447055, I)
Affinity DataKi:  1nMAssay Description:The potency of inhibition of compound I and compound II on prostaglandin F2α receptor was assessed by analyzing the affinity of these compounds...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410625(CHEMBL2113201)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410634(CHEMBL2113189)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM50313357(3-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...)
Affinity DataKi:  2nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410622(CHEMBL2113203)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410634(CHEMBL2113189)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM50313351(6-(dipropylamino)-N-(1H-indazol-5-yl)pyrimidine-4-...)
Affinity DataKi:  3nM ΔG°:  -45.2kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410619(CHEMBL2113208)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM183667(US9150519, 1-55)
Affinity DataKi:  3.20nM ΔG°:  -45.1kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86209(Atosiban | CAS_90779-69-4 | NSC_0)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21599(2-{5-chloro-1'-[(3-methyl-5-phenyl-1,2-oxazol-4-yl...)
Affinity DataKi:  3.80nM EC50:  19nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410640(CHEMBL2113198)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410623(CHEMBL2113179)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410625(CHEMBL2113201)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Mus musculus (mouse))
Merck Serono

LigandPNGBDBM21610(2-[(3R)-5-chloro-1'-[(5-chloro-2-fluorophenyl)meth...)
Affinity DataKi:  5nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21595(2-{5-chloro-1'-[(3-methyl-5-phenyl-1,2-oxazol-4-yl...)
Affinity DataKi:  5.30nM EC50:  23nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21610(2-[(3R)-5-chloro-1'-[(5-chloro-2-fluorophenyl)meth...)
Affinity DataKi:  5.30nM EC50:  66nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM244800(US9447055, II)
Affinity DataKi:  6nMAssay Description:The potency of inhibition of compound I and compound II on prostaglandin F2α receptor was assessed by analyzing the affinity of these compounds...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM50313358(3-(4-(6-((cyclopropylmethyl)(propyl)amino)pyrimidi...)
Affinity DataKi:  6nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM183686(US9150519, 1-84)
Affinity DataKi:  7nM ΔG°:  -43.3kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410621(CHEMBL2113177)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410635(CHEMBL2113211)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM183668(US9150519, 1-56)
Affinity DataKi:  7nM ΔG°:  -43.3kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21594(2-{5-chloro-1'-[(5-methyl-3-phenyl-1,2-oxazol-4-yl...)
Affinity DataKi:  7.60nM EC50:  21nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM50313359(4-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...)
Affinity DataKi:  8nM ΔG°:  -43.0kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410616(CHEMBL2113185)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM183701(US9150519, 1-100)
Affinity DataKi:  8nM ΔG°:  -43.0kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410638(CHEMBL2113207)
Affinity DataKi:  8.70nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM183699(US9150519, 1-97)
Affinity DataKi:  9nM ΔG°:  -42.7kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM50313363(3-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...)
Affinity DataKi:  9nM ΔG°:  -42.7kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM183676(US9150519, 1-69)
Affinity DataKi:  10nM ΔG°:  -42.4kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410630(CHEMBL2113209)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21579(2-{5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1...)
Affinity DataKi:  10nM EC50:  48nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410619(CHEMBL2113208)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21596(2-{5-chloro-1'-[(4-methoxy-3,5-dimethylpyridin-2-y...)
Affinity DataKi:  12nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Serono

US Patent
LigandPNGBDBM50313361(2-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...)
Affinity DataKi:  12nM ΔG°:  -42.0kJ/molepH: 7.4 T: 2°CAssay Description:Membranes were prepared from CHO cells expressing S1P1 or S1P3 for use in ligand and 35S-GTPgammaS binding studies. Cells were suspended in 50 mM TRI...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Serono

LigandPNGBDBM21611(2-[(3S)-5-chloro-1'-[(5-chloro-2-fluorophenyl)meth...)
Affinity DataKi:  13nMAssay Description:A scintillation proximity assay was used for radioligand competition and saturation binding assays. Nonspecific binding was determined in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50178153(4-ethoxy-N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50178186(CHEMBL372122 | N-(4-chlorophenyl)-4-ethoxy-N-{2-[(...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410622(CHEMBL2113203)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50326713((2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methox...)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410637(CHEMBL2113210)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50178209(CHEMBL371223 | N-(4-chlorophenyl)-3,4-dimethoxy-N-...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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