Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 885nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat DAT-mediated dopamine reuptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat DAT-mediated dopamine reuptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat NET-mediated norepinephrine reuptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat NET-mediated norepinephrine reuptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of rat DAT-mediated dopamine reuptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of rat SERT-mediated serotonin reuptakeMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Cephalon (France)
Curated by ChEMBL
Cephalon (France)
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of rat SERT-mediated serotonin reuptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A5More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A5More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 6.39E+4nMAssay Description:Inhibition of rat NET-mediated norepinephrine reuptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair