Compile Data Set for Download or QSAR
maximum 50k data
Found 56 with Last Name = 'schwerdt' and Initial = 'jh'
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175843(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175828(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175833(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175843(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177371(2-((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)e...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177376(4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177385((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177387((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177379((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177386(4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177384((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177383(4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177380((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175833(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175828(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175851(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-p...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175836(CHEMBL200643 | N-(3-(4-((1H-imidazol-4-yl)methyl)p...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175827(4-((1H-imidazol-4-yl)methyl)-1-heptylpiperidine | ...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175846(4-((1H-imidazol-4-yl)methyl)-1-(3-(3-chlorophenoxy...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177375((R)-4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175829(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-c...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175831(CHEMBL373263 | methyl 4-(3-(4-((1H-imidazol-4-yl)m...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175830(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177370((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177374((R)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175839(4-((1H-imidazol-4-yl)methyl)-1-(3-phenoxypropyl)pi...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177378(4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175837(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-p...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175838(4-((1H-imidazol-4-yl)methyl)-1-(4-phenylbutyl)pipe...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177377((R)-4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175857(4-((1H-imidazol-4-yl)methyl)-1-(4-(4-chlorophenyl)...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177382(4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-(4...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175856(CHEMBL200519 | N-(2-(4-((1H-imidazol-4-yl)methyl)p...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175832(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-4-p...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175845(CHEMBL200806 | N-(3-(4-((1H-imidazol-4-yl)methyl)p...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175844(4-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175855(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)hept...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175850(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175848(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175826(4-((1H-imidazol-4-yl)methyl)-1-(3-(phenylsulfonyl)...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175854(5-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177372((S)-4-(((R)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175847(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175835(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175841(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177373((S)-4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175849(2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177381((R)-4-(((S)-1-(3,5-bis(trifluoromethyl)phenyl)etho...)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]-Sar-Met Substance P from recombinant human NK1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175842(4-((1H-imidazol-4-yl)methyl)-N-(4-chlorophenyl)pip...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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