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Found 88 with Last Name = 'scriba' and Initial = 'gk'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...)
Affinity DataKi:  2.75nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...)
Affinity DataKi:  18.6nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  18.6nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181460(1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-d...)
Affinity DataKi:  243nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181463(1,3-bis(4-chlorophenyl)-5-phenylimidazolidine-2,4-...)
Affinity DataKi:  247nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181460(1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-d...)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181463(1,3-bis(4-chlorophenyl)-5-phenylimidazolidine-2,4-...)
Affinity DataKi:  353nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177155(1-(bis(4-bromophenyl)methyl)-3-(4-bromophenyl)urea...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164429(3-Allyl-5,5-bis-(4-iodo-phenyl)-2-thioxo-imidazoli...)
Affinity DataKi:  589nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177162(1-[bis(4-bromophenyl)methyl]-3-(4-chlorophenyl)-ur...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181462(1,3-bis(3-iodophenyl)-5-phenyl-2-thioxoimidazolidi...)
Affinity DataKi:  692nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164432(3-Butyl-5,5-bis-(4-iodo-phenyl)-2-thioxo-imidazoli...)
Affinity DataKi:  724nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177160(1-[bis(4-iodophenyl)methyl]-3-(4-bromophenyl)urea ...)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164431(3-Allyl-5,5-bis-(4-bromo-phenyl)-2-thioxo-imidazol...)
Affinity DataKi:  871nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181458(5-(4-bromophenyl)-1,3-bis(4-chlorophenyl)imidazoli...)
Affinity DataKi:  905nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164441(3-Benzyl-5,5-bis-(4-bromo-phenyl)-2-thioxo-imidazo...)
Affinity DataKi:  993nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177159(1-[bis(4-chlorophenyl)methyl]-3-(4-chlorophenyl)- ...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177163(1-(bis(4-chlorophenyl)methyl)-3-(4-bromophenyl)ure...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164442(5,5-Bis-(4-bromo-phenyl)-3-butyl-2-thioxo-imidazol...)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181461(1,3-bis(4-bromophenyl)-5-phenyl-2-thioxoimidazolid...)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177164(1-[bis(4-bromophenyl)methyl]-3-(4-chlorophenyl)thi...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164439(3-Allyl-5,5-bis-(4-iodo-phenyl)-imidazolidine-2,4-...)
Affinity DataKi:  1.74E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181458(5-(4-bromophenyl)-1,3-bis(4-chlorophenyl)imidazoli...)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164433(5,5-Bis-(4-bromo-phenyl)-3-isobutyl-2-thioxo-imida...)
Affinity DataKi:  1.78E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177158(1-[bis(4-bromophenyl)methyl]-3-phenylthiourea | CH...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164430(3-Butyl-5,5-bis-(4-iodo-phenyl)-imidazolidine-2,4-...)
Affinity DataKi:  1.82E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181459(1,3,5-tris(4-chlorophenyl)imidazolidine-2,4-dione ...)
Affinity DataKi:  1.88E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177157(1-[bis(4-chlorophenyl)methyl]-3-(4-chlorophenyl)th...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181466(1,3-bis(4,3-dichlorophenyl)-5-phenyl-2-thioxoimida...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164438(5,5-Bis-(4-chloro-phenyl)-3-isobutyl-2-thioxo-imid...)
Affinity DataKi:  2.09E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181469(1,3-bis(3-chlorophenyl)-5-phenylimidazolidine-2,4-...)
Affinity DataKi:  2.11E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181456(1,3-bis(4-chlorophenyl)-5-phenyl-2-thioxoimidazoli...)
Affinity DataKi:  2.16E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164440(3-Benzyl-5,5-bis-(4-chloro-phenyl)-2-thioxo-imidaz...)
Affinity DataKi:  2.19E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164428(5,5-Bis-(4-bromo-phenyl)-3-ethyl-2-thioxo-imidazol...)
Affinity DataKi:  2.19E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181459(1,3,5-tris(4-chlorophenyl)imidazolidine-2,4-dione ...)
Affinity DataKi:  2.62E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177156(5,5'-bis(4-bromophenyl)-3-(4-chlorophenyl)-2-thiox...)
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177167(1-(bis(4-bromophenyl)methyl)-3-phenylurea | CHEMBL...)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177161(1-[bis(4-chlorophenyl)methyl]-3-phenylthiourea | C...)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50181455(1,3-bis(3-chlorophenyl)-5-(4-chlorophenyl)imidazol...)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50177166(5,5'-bis(4-bromophenyl)-3-phenyl-2-thioxoimidazoli...)
Affinity DataKi:  3.45E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164443(3-Benzyl-5,5-bis-(4-bromo-phenyl)-imidazolidine-2,...)
Affinity DataKi:  3.47E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164437(5,5-Bis-(4-bromo-phenyl)-3-isopropyl-2-thioxo-imid...)
Affinity DataKi:  3.63E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164435(5,5-Bis-(4-chloro-phenyl)-3-phenethyl-2-thioxo-imi...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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