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Found 100 with Last Name = 'scrima' and Initial = 'm'
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50430016(CHEMBL2335444)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant full length CAMK2alpha (unknown origin) using autocamtide-2 as substrate assessed as incorporation of 32P after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50430015(CHEMBL2335442)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant full length CAMK2alpha (unknown origin) using autocamtide-2 as substrate assessed as incorporation of 32P after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50430014(CHEMBL2335479)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant full length CAMK2alpha (unknown origin) using autocamtide-2 as substrate assessed as incorporation of 32P after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50024797(CHEBI:60283 | CHEMBL1163500 | N6-Isopentenyladenos...)
Affinity DataKd:  1.21E+6nMAssay Description:Binding affinity to FPPS (unknown origin) expressed in Escherichia coli BL21(DEscherichia ) assessed as binding constant of proton H14-H15 of isopent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50024797(CHEBI:60283 | CHEMBL1163500 | N6-Isopentenyladenos...)
Affinity DataKd:  5.50E+5nMAssay Description:Binding affinity to FPPS (unknown origin) expressed in Escherichia coli BL21(DEscherichia ) assessed as binding constant of proton H11 of isopentenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50024797(CHEBI:60283 | CHEMBL1163500 | N6-Isopentenyladenos...)
Affinity DataKd:  2.21E+6nMAssay Description:Binding affinity to FPPS (unknown origin) expressed in Escherichia coli BL21(DEscherichia ) assessed as binding constant of proton H12 of isopentenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50024797(CHEBI:60283 | CHEMBL1163500 | N6-Isopentenyladenos...)
Affinity DataKd:  2.02E+6nMAssay Description:Binding affinity to FPPS (unknown origin) expressed in Escherichia coli BL21(DEscherichia ) assessed as binding constant of proton H2/H8 of purine ri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.190nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.0700nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031470(CHEMBL3358551)
Affinity DataEC50:  0.150nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031471(CHEMBL3358550)
Affinity DataEC50:  0.150nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.0450nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031476(CHEMBL3358548)
Affinity DataEC50:  1.90nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031477(CHEMBL3358547)
Affinity DataEC50:  1.80nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.0420nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.340nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031487(CHEMBL3358543)
Affinity DataEC50:  1.90nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.0510nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031489(CHEMBL3352878)
Affinity DataEC50:  0.230nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031490(CHEMBL3358540)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031492(CHEMBL3358539)
Affinity DataEC50:  0.0860nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031493(CHEMBL3358538)
Affinity DataEC50:  5nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)
Affinity DataEC50:  1.90nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031495(CHEMBL3358536)
Affinity DataEC50:  0.180nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031496(CHEMBL3358535)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031497(CHEMBL3358534)
Affinity DataEC50:  5.30nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031498(CHEMBL3358533)
Affinity DataEC50:  3.20nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.0600nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.0670nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031470(CHEMBL3358551)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031471(CHEMBL3358550)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.0480nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031476(CHEMBL3358548)
Affinity DataEC50:  0.850nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031477(CHEMBL3358547)
Affinity DataEC50:  0.580nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.0510nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.220nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031487(CHEMBL3358543)
Affinity DataEC50:  1.60nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031499(CHEMBL3358542)
Affinity DataEC50:  0.310nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031500(CHEMBL2372859)
Affinity DataEC50:  0.210nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.0580nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031489(CHEMBL3352878)
Affinity DataEC50:  0.290nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031490(CHEMBL3358540)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031492(CHEMBL3358539)
Affinity DataEC50:  0.0980nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031493(CHEMBL3358538)
Affinity DataEC50:  2.20nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)
Affinity DataEC50:  0.810nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031495(CHEMBL3358536)
Affinity DataEC50:  0.190nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031496(CHEMBL3358535)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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