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Found 86 with Last Name = 'sekiyama' and Initial = 'n'
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:The compound was evaluated for agonist to competitive inhibition of radioligand ([3H]- CPP ) at Ionotropic Excitatory Amino acid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  1.20E+4nMAssay Description:Effect on Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)
Affinity DataEC50:  1.40E+5nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >5.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)
Affinity DataEC50: >3.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  4.00E+3nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50:  5.80E+4nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060718((R)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  5.40E+6nMAssay Description:Effect on Metabotropic glutamate receptor 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  910nMAssay Description:Effect on Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  2.52E+5nMAssay Description:Effect on Metabotropic glutamate receptor 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  4.40E+3nMAssay Description:Effect on Metabotropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  9.00E+3nMAssay Description:Effect on Metabotropic glutamate receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)
Affinity DataEC50:  3.50E+4nMAssay Description:Effect on Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052553((2S)-2-aminohexanedioic acid | (S)-2-aminohexanedi...)
Affinity DataEC50: >3.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  2.00E+4nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  570nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052551(2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyr...)
Affinity DataEC50:  8.20E+4nMAssay Description:Effect on Metabotropic glutamate receptor 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >5.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060719((S)-2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-b...)
Affinity DataEC50: >1.00E+6nMAssay Description:Effect on Metabotropic glutamate receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM17662((2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl...)
Affinity DataEC50:  2.20E+5nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM31174(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50052549(2-Amino-heptanedioic acid | CHEMBL111050)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataEC50:  8.50E+3nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonistic activity at mGlu6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM85356((S)-2-Aminoadipic acid | CAS_542-32-5)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004852(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM31174(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonistic activity at mGlu2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026947((R)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)-p...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu1-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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