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Found 71 with Last Name = 'sergejew' and Initial = 't'
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035208(1-Pyridin-4-yl-1a,2,3,7b-tetrahydro-1H-cyclopropa[...)
Affinity DataIC50:  66nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035206(4-(5-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049763(2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...)
Affinity DataIC50:  170nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035209(4-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  185nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049763(2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  265nMAssay Description:In vitro inhibition of rat ovarian microsomal Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035211(1-Pyridin-4-yl-1a,2,3,7b-tetrahydro-1H-cyclopropa[...)
Affinity DataIC50:  330nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035209(4-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  370nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035213(4-(6-Methoxy-1-methyl-1a,2,3,7b-tetrahydro-1H-cycl...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM8611(4-{5H,6H,7H,8H-imidazo[1,5-a]pyridin-5-yl}benzonit...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049774(5-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035205(4-(5-Bromo-6-methoxy-1a,2,3,7b-tetrahydro-1H-cyclo...)
Affinity DataIC50:  920nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035205(4-(5-Bromo-6-methoxy-1a,2,3,7b-tetrahydro-1H-cyclo...)
Affinity DataIC50:  920nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049777(2-[1-Thiazol-5-yl-meth-(E)-ylidene]-3,4-dihydro-2H...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035209(4-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035212(4-(4-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  3.35E+3nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035210(4-(7-Bromo-4-methoxy-1a,2,3,7b-tetrahydro-1H-cyclo...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50009605(2-(pyridin-4-ylmethylene)-3,4-dihydronaphthalen-1(...)
Affinity DataIC50:  4.60E+3nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035207(1-(pyridin-4-yl)-1a,2,3,7b-tetrahydro-1H-cycloprop...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  6.20E+3nMAssay Description:In vitro inhibition of rat ovarian microsomal Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035208(1-Pyridin-4-yl-1a,2,3,7b-tetrahydro-1H-cyclopropa[...)
Affinity DataIC50:  7.00E+3nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049765(2-[1-Pyridin-3-yl-meth-(E)-ylidene]-3,4-dihydro-2H...)
Affinity DataIC50:  9.20E+3nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049768(2-[1-Pyrazin-2-yl-meth-(E)-ylidene]-3,4-dihydro-2H...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50378780((S)-VOROZOLE)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50009605(2-(pyridin-4-ylmethylene)-3,4-dihydronaphthalen-1(...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049776(3-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  1.30E+4nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049766(1-Phenyl-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]naph...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049778(2-[1-(2H-Pyrazol-3-yl)-meth-(E)-ylidene]-3,4-dihyd...)
Affinity DataIC50:  1.80E+4nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of Human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049762(3-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049778(2-[1-(2H-Pyrazol-3-yl)-meth-(E)-ylidene]-3,4-dihyd...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid 17-alpha-hydroxylase/17,20 lyase(Rattus norvegicus (Rat))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049777(2-[1-Thiazol-5-yl-meth-(E)-ylidene]-3,4-dihydro-2H...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro inhibitory activity against Steroidgenic Cytochrome P450 17 alpha using rat testicular microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049764(2-[1-Pyridazin-3-yl-meth-(E)-ylidene]-3,4-dihydro-...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049776(3-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049775(2-(Hydroxy-pyrimidin-4-yl-methyl)-3,4-dihydro-2H-n...)
Affinity DataIC50:  2.70E+4nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B1, mitochondrial(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro inhibition of ACTH-stimulated corticosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B1, mitochondrial(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035204(4-(6-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro inhibition of ACTH-stimulated corticosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid 17-alpha-hydroxylase/17,20 lyase(Rattus norvegicus (Rat))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049763(2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...)
Affinity DataIC50:  3.10E+4nMAssay Description:In vitro inhibitory activity against Steroidgenic Cytochrome P450 17 alpha using rat testicular microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid 17-alpha-hydroxylase/17,20 lyase(Rattus norvegicus (Rat))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035209(4-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  3.60E+4nMAssay Description:In vitro inhibitory activity against Steroidgenic Cytochrome P450 17 alpha using rat testicular microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid 17-alpha-hydroxylase/17,20 lyase(Rattus norvegicus (Rat))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50009605(2-(pyridin-4-ylmethylene)-3,4-dihydronaphthalen-1(...)
Affinity DataIC50:  3.70E+4nMAssay Description:In vitro inhibitory activity against Steroidgenic Cytochrome P450 17 alpha using rat testicular microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049768(2-[1-Pyrazin-2-yl-meth-(E)-ylidene]-3,4-dihydro-2H...)
Affinity DataIC50:  3.80E+4nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049763(2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid 17-alpha-hydroxylase/17,20 lyase(Rattus norvegicus (Rat))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049765(2-[1-Pyridin-3-yl-meth-(E)-ylidene]-3,4-dihydro-2H...)
Affinity DataIC50:  4.80E+4nMAssay Description:In vitro inhibitory activity against Steroidgenic Cytochrome P450 17 alpha using rat testicular microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Rattus norvegicus)
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibition of ACTH-stimulated aldosterone biosynthesis in rat adrenal slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
UniversitäT Des Saarlandes

Curated by ChEMBL
LigandPNGBDBM50049762(3-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  5.10E+4nMAssay Description:In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
UniversitäT De Saarlandes

Curated by ChEMBL
LigandPNGBDBM50035209(4-(1a,2,3,7b-Tetrahydro-1H-cyclopropa[a]naphthalen...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibitory activity against Steroidgenic Cytochrome P450 C18 using Bovine adrenal mitochondria.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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